Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 74
TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159110(US9682967, 6)
Affinity DataIC50: 4.00E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445041(CHEMBL3098768 | US9682967, 46 | US10195186, Exampl...)
Affinity DataKi:  84nM IC50: 88nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445042(CHEMBL3098767 | US9682967, 7 | US10195186, Example...)
Affinity DataKi:  162nM IC50: 170nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159232(US9682967, 45 | US10195186, Example 47)
Affinity DataKi:  190nM IC50: 200nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Mouse)
H. Lundbeck

US Patent
LigandPNGBDBM50445054(CHEMBL3098745 | US9682967, 1 | US10195186, Example...)
Affinity DataKi:  210nM IC50: 220nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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PDB3D3D Structure (crystal)
TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159140(US9682967, 18 | US10195186, Example 18)
Affinity DataKi:  229nM IC50: 240nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159226(US9682967, 44 | US10195186, Example 46)
Affinity DataKi:  286nM IC50: 300nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159139(US9682967, 17 | US10195186, Example 17)
Affinity DataKi:  343nM IC50: 360nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159138(US9682967, 16 | US10195186, Example 16)
Affinity DataKi:  343nM IC50: 360nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445054(CHEMBL3098745 | US9682967, 1 | US10195186, Example...)
Affinity DataKi:  429nM IC50: 450nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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PDB3D3D Structure (crystal)
TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159123(US9682967, 11 | US10195186, Example 11)
Affinity DataKi:  457nM IC50: 480nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159129(US9682967, 13 | US10195186, Example 13)
Affinity DataKi:  457nM IC50: 480nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445044(CHEMBL3098765 | US9682967, 34 | US10195186, Exampl...)
Affinity DataKi:  467nM IC50: 490nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159154(US9682967, 23 | US10195186, Example 23)
Affinity DataKi:  543nM IC50: 570nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159285(US9682967, 50)
Affinity DataKi:  599nM IC50: 620nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159286(US9682967, 51)
Affinity DataKi:  614nM IC50: 640nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159121(US9682967, 9 | US10195186, Example 9)
Affinity DataKi:  667nM IC50: 700nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159189(US9682967, 36 | US10195186, Example 38)
Affinity DataKi:  714nM IC50: 750nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159272(US9682967, 48 | US10195186, Example 50)
Affinity DataKi:  721nM IC50: 760nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159273(US9682967, 49 | US10195186, Example 51)
Affinity DataKi:  734nM IC50: 750nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445051(CHEMBL3098752 | US9682967, 5 | US10195186, Example...)
Affinity DataKi:  790nM IC50: 830nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159181(US9682967, 33 | US10195186, Example 35)
Affinity DataKi:  924nM IC50: 970nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159146(US9682967, 20 | US10195186, Example 20)
Affinity DataKi:  943nM IC50: 990nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159117(US9682967, 8 | US10195186, Example 8)
Affinity DataKi:  952nM IC50: 1.00E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445055(CHEMBL3098744 | US9682967, 43 | US10195186, Exampl...)
Affinity DataKi:  1.05E+3nM IC50: 1.10E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445058(CHEMBL3098741 | US9682967, 2 | US10195186, Example...)
Affinity DataKi:  1.14E+3nM IC50: 1.20E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159271(US9682967, 47 | US10195186, Example 49)
Affinity DataKi:  1.14E+3nM IC50: 1.20E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445043(CHEMBL3098766 | US9682967, 37 | US10195186, Exampl...)
Affinity DataKi:  1.24E+3nM IC50: 1.30E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159169(US9682967, 29 | US10195186, Example 30)
Affinity DataKi:  1.24E+3nM IC50: 1.30E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445057(CHEMBL3098742 | US9682967, 4 | US10195186, Example...)
Affinity DataKi:  1.33E+3nM IC50: 1.40E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445047(CHEMBL3098760 | US9682967, 22 | US10195186, Exampl...)
Affinity DataKi:  1.52E+3nM IC50: 1.60E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159199(US9682967, 38 | US10195186, Example 40)
Affinity DataKi:  1.52E+3nM IC50: 1.60E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159143(US9682967, 19 | US10195186, Example 19)
Affinity DataKi:  1.62E+3nM IC50: 1.70E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445045(CHEMBL3098764 | US9682967, 25 | US10195186, Exampl...)
Affinity DataKi:  1.71E+3nM IC50: 1.80E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159126(US9682967, 12 | US10195186, Example 12)
Affinity DataKi:  1.71E+3nM IC50: 1.80E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159188(US9682967, 35 | US10195186, Example 37)
Affinity DataKi:  1.91E+3nM IC50: 2.00E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159172(US9682967, 30 | US10195186, Example 32)
Affinity DataKi:  2.00E+3nM IC50: 2.10E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159122(US9682967, 10 | US10195186, Example 10)
Affinity DataKi:  2.10E+3nM IC50: 2.20E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445046(CHEMBL3098761 | US9682967, 24 | US10195186, Exampl...)
Affinity DataKi:  2.29E+3nM IC50: 2.40E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159178(US9682967, 32 | US10195186, Example 34)
Affinity DataKi:  3.05E+3nM IC50: 3.20E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445050(CHEMBL3098753 | US9682967, 15 | US10195186, Exampl...)
Affinity DataKi:  3.24E+3nM IC50: 3.40E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159210(US9682967, 41 | US10195186, Example 43)
Affinity DataKi:  3.43E+3nM IC50: 3.60E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159166(US9682967, 28 | US10195186, Example 29)
Affinity DataKi:  3.43E+3nM IC50: 3.60E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445048(CHEMBL3098759 | US9682967, 21 | US10195186, Exampl...)
Affinity DataKi:  3.43E+3nM IC50: 3.60E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159134(US9682967, 14 | US10195186, Example 14)
Affinity DataKi:  4.00E+3nM IC50: 4.20E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159206(US9682967, 40 | US10195186, Example 42)
Affinity DataKi:  4.57E+3nM IC50: 4.80E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159213(US9682967, 42 | US10195186, Example 44)
Affinity DataKi:  4.95E+3nM IC50: 5.20E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159162(US9682967, 26 | US10195186, Example 26)
Affinity DataKi:  5.24E+3nM IC50: 5.50E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50445056(CHEMBL3098743 | US9682967, 3 | US10195186, Example...)
Affinity DataKi:  6.10E+3nM IC50: 6.40E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
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TargetSortilin(Human)
H. Lundbeck

US Patent
LigandPNGBDBM159202(US9682967, 39 | US10195186, Example 41)
Affinity DataKi:  7.14E+3nM IC50: 7.50E+3nMpH: 7.4Assay Description:The Sortilin assay was performed in total volume of 40 ul in 50 mM HEPES pH 7.4 assay buffer containing 100 mM NaCl, 2.0 mM CaCl2, 0.1% BSA and 0.1% ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
Go to US Patent