Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 139
LigandPNGBDBM189846(US9670194, Ex. 65 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 2nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188124(US9670194, Ex. 3 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50: 2nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188116(US9670194, Ex. 1 (S)-2-(1-((6-amino-5-(5-methyl-1,...)
Affinity DataIC50: 3nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189408(US9670194, Ex. 41 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 5nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189403(US9670194, Ex. 37 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 6nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189838(US9670194, Ex. 57 (S)-2-(1-((6-amino-5-(3-isopropy...)
Affinity DataIC50: 6nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189845(US9670194, Ex. 64 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 8nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188145(US9670194, Ex. 4 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50: 8nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189837(US9670194, Ex. 56 (S)-2-(1-((6-amino-5-(3-ethyl-1,...)
Affinity DataIC50: 9nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189405(US9670194, Ex. 39 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 11nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189404(US9670194, Ex. 38 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 12nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189306(US9670194, Ex. 34 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 12nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189298(US9670194, Ex. 27 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 13nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189832(US9670194, Ex. 52 (S)-2-(1-((6-amino-5-(4-methylox...)
Affinity DataIC50: 15nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189303(US9670194, Ex. 31 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 18nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189844(US9670194, Ex. 63 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 18nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188473(US9670194, Ex. 21 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 19nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188332(US9670194, Ex. 14 (S)-2-(1-((6-amino-5-(isoxazol-3...)
Affinity DataIC50: 20nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189840(US9670194, Ex. 59 (S)-2-(1-((6-amino-5-(5-isopropy...)
Affinity DataIC50: 20nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188474(US9670194, Ex. 22 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 26nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188117(US9670194, Ex. 2 (S)-2-(1-((6-amino-5-(5-methyl-1,...)
Affinity DataIC50: 33nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189408(US9670194, Ex. 41 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 35nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189843(US9670194, Ex. 62 2-((S)-1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 37nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189846(US9670194, Ex. 65 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 37nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189842(US9670194, Ex. 61 (S)-2-(1-((6-amino-5-(5-ethyl-1,...)
Affinity DataIC50: 44nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188330(US9670194, Ex. 12 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 48nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188338(US9670194, Ex. 20 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 49nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188475(US9670194, Ex. 23 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 52nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188124(US9670194, Ex. 3 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50: 66nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189305(US9670194, Ex. 33 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 67nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189304(US9670194, Ex. 32 (S)-2-(1-((6-amino-5-(1-methyl-1...)
Affinity DataIC50: 70nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189406(US9670194, Ex. 40 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 93nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188324(US9670194, Ex. 6 2-((S)-1((6-amino-5-((S)-4-methyl...)
Affinity DataIC50: 99nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189845(US9670194, Ex. 64 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 112nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188145(US9670194, Ex. 4 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50: 113nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189829(US9670194, Ex. 51 (S)-2-(1-((6-amino-5-(1-methyl-1...)
Affinity DataIC50: 135nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188124(US9670194, Ex. 3 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50: 142nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189846(US9670194, Ex. 65 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 154nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188117(US9670194, Ex. 2 (S)-2-(1-((6-amino-5-(5-methyl-1,...)
Affinity DataIC50: 168nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189833(US9670194, Ex. 53 (S)-2-(1-((6-amino-5-(1-methyl-1...)
Affinity DataIC50: 239nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188325(US9670194, Ex. 7 (S)-2-(1-((6-amino-5-(5-methyloxa...)
Affinity DataIC50: 246nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188145(US9670194, Ex. 4 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50: 258nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189408(US9670194, Ex. 41 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 261nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189844(US9670194, Ex. 63 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 269nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189295(US9670194, Ex. 25 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 298nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189795(US9670194, Ex. 44 (S)-2-(1-((6-amino-5-(1-methyl-1...)
Affinity DataIC50: 358nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188116(US9670194, Ex. 1 (S)-2-(1-((6-amino-5-(5-methyl-1,...)
Affinity DataIC50: 384nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM188124(US9670194, Ex. 3 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50: 442nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189405(US9670194, Ex. 39 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50: 502nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM189845(US9670194, Ex. 64 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50: 674nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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