Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 853
LigandPNGBDBM294260(US9586945, 15b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294276(US9586945, 27 | Cis-N-(1-(4-benzyl-7-fluoro-3-(met...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294256(US9586945, 13 | Cis-N-(1-(4-benzyl-3-(methylamino)...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294271(US9586945, 22 | US9586945, 23* | Cis-N-(1-(4-benz...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294270(US9586945, 21)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294268(US9586945, 19b | trans-N-(1-(4-benzyl-7-fluoro-3-...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294267(US9586945, 19a | Cis-N-(1-(4-benzyl-7-fluoro-3-(m...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294266(US9586945, 18b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294265(US9586945, 18a | Cis-N-(1-(4-benzyl-7-fluoro-3-(me...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294264(US9586945, 17b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294263(US9586945, 17a | Cis-N-(1-(4-benzyl-7-fluoro-3-(m...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294262(US9586945, 16b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294261(US9586945, 16a | Cis-N-(1-(4-benzyl-7-fluoro-3-(m...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294259(US9586945, 15a | Cis-N-(1-(4-benzyl-7-fluoro-3-(m...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294244(US9586945, 1 | N-[1-[3-(azetidin-1-yl)-4-benzyl-c...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294256(US9586945, 13 | Cis-N-(1-(4-benzyl-3-(methylamino)...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294254(US9586945, 11 | Cis-N-(1-(4-benzyl-3-(methylamino)...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294249(US9586945, 6 | Cis-N-(1-(3-(azetidin-1-yl)-4-benzy...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294250(US9586945, 7 | Cis-N-(1-(3-(azetidin-1-yl)-4-benzy...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294275(US9586945, 26 | Cis-1-(4-benzyl-7-fluoro-6-(3-(5-f...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294276(US9586945, 27 | Cis-N-(1-(4-benzyl-7-fluoro-3-(met...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294246(US9586945, 3 | Cis-N-(1-(3-(azetidin-1-yl)-4-benzy...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294278(US9586945, 29 | Cis-N-(1-(4-benzyl-3-(propylamino)...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294247(US9586945, 4 | Cis-N-(1-(3-(azetidin-1-yl)-4-benzy...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294248(US9586945, 5 | Cis-N-(1-(3-(azetidin-1-yl)-4-benzy...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294269(US9586945, 20)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294258(US9586945, 14b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294279(US9586945, 30 | Cis-N-(1-(4-benzyl-3-(diethylamino...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294253(US9586945, 10 | Cis-N-(1-(3-(azetidin-1-yl)-4-benz...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294255(US9586945, 12 | Cis-N-(1-(-4-benzyl-3-(methylamino...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294257(US9586945, 14a | Cis-N-(1-(4-benzyl-7-fluoro-3-(me...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294280(US9586945, 31 | Cis-N-(1-(4-benzyl-3-((cyclopropyl...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294281(US9586945, 32* | Cis-N-(1-(4-benzyl-3-(cyclobutyl...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294274(US9586945, 25 | Cis-N-(1-(4-benzyl-3-(methylamino)...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294271(US9586945, 22 | US9586945, 23* | Cis-N-(1-(4-benz...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294252(US9586945, 9 | Cis-N-(1-(3-(azetidin-1-yl)-4-benzy...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294251(US9586945, 8 | Cis-N-(1-(3-(azetidin-1-yl)-4-benzy...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM294245(US9586945, 2 | Cis-N-(1-(3-(azetidin-1-yl)-4-benzy...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
In DepthDetails
US Patent