Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 210
TargetEstrogen receptor beta(Human)
Donesta Bioscience

US Patent
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataKi:  0.0150nMpH: 7.5Assay Description:The method employed was adapted from the scientific literature and described in detail by Osbourn et al. (1993, Biochemistry, 32, 6229-6236). Recombi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEstrogen receptor beta(Human)
Donesta Bioscience

US Patent
LigandPNGBDBM158504(US9034854, EE | US9561238, EE | US9040509, EE)
Affinity DataKi:  0.0250nMpH: 7.5Assay Description:The method employed was adapted from the scientific literature and described in detail by Osbourn et al. (1993, Biochemistry, 32, 6229-6236). Recombi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEstrogen receptor(Human)
Donesta Bioscience

US Patent
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataKi:  0.210nMpH: 7.5Assay Description:The method employed was adapted from the scientific literature and described in detail by Osbourn et al. (1993, Biochemistry, 32, 6229-6236). Recombi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEstrogen receptor(Human)
Donesta Bioscience

US Patent
LigandPNGBDBM158504(US9034854, EE | US9561238, EE | US9040509, EE)
Affinity DataKi:  0.230nMpH: 7.5Assay Description:The method employed was adapted from the scientific literature and described in detail by Osbourn et al. (1993, Biochemistry, 32, 6229-6236). Recombi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEstrogen receptor(Human)
Donesta Bioscience

US Patent
LigandPNGBDBM158505(US9034854, E4 | US9561238, E4 | US9040509, E4)
Affinity DataKi:  4.90nMpH: 7.5Assay Description:The method employed was adapted from the scientific literature and described in detail by Osbourn et al. (1993, Biochemistry, 32, 6229-6236). Recombi...More data for this Ligand-Target Pair
In DepthDetails
US Patent
PDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Human)
Donesta Bioscience

US Patent
LigandPNGBDBM158505(US9034854, E4 | US9561238, E4 | US9040509, E4)
Affinity DataKi:  19nMpH: 7.5Assay Description:The method employed was adapted from the scientific literature and described in detail by Osbourn et al. (1993, Biochemistry, 32, 6229-6236). Recombi...More data for this Ligand-Target Pair
In DepthDetails
US Patent