Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 212
LigandPNGBDBM228153((S)-5-(4-morpholino-5a,6,8,9-tetrahydro-5H- pyrimi...)
Affinity DataIC50: 98.1nMpH: 7.5Assay Description:N-terminally His-tagged PI3K alpha (Cat. No. PV4789; 0.49 mg/ml), Alexa Fluor 647 labeled kinase Tracer 314 (Cat. No. PV6087), Biotin anti-His Tag an...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM228157((S)-5-(2-morpholino-5a,6,8,9-tetrahydro-5H- pyrimi...)
Affinity DataIC50: 383nMpH: 7.5Assay Description:N-terminally His-tagged PI3K alpha (Cat. No. PV4789; 0.49 mg/ml), Alexa Fluor 647 labeled kinase Tracer 314 (Cat. No. PV6087), Biotin anti-His Tag an...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM228130((R)-5-(4-morpholino-5a,6,8,9-tetrahydro-5H- pyrimi...)
Affinity DataIC50: 390nMpH: 7.5Assay Description:N-terminally His-tagged PI3K alpha (Cat. No. PV4789; 0.49 mg/ml), Alexa Fluor 647 labeled kinase Tracer 314 (Cat. No. PV6087), Biotin anti-His Tag an...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM228155((R)-5-(2-morpholino-5a,6,8,9-tetrahydro-5H- pyrimi...)
Affinity DataIC50: 2.62E+3nMpH: 7.5Assay Description:N-terminally His-tagged PI3K alpha (Cat. No. PV4789; 0.49 mg/ml), Alexa Fluor 647 labeled kinase Tracer 314 (Cat. No. PV6087), Biotin anti-His Tag an...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM228154((S)-5-(4-morpholino-5a,6,8,9-tetrahydro-5H- pyrimi...)
Affinity DataKi:  8nM IC50: 76nMpH: 7.5Assay Description:N-terminally His-tagged PI3K alpha (Cat. No. PV4789; 0.49 mg/ml), Alexa Fluor 647 labeled kinase Tracer 314 (Cat. No. PV6087), Biotin anti-His Tag an...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM228156((R)-5-(2-morpholino-5a,6,8,9-tetrahydro-5H- pyrimi...)
Affinity DataKi:  23nM IC50: 231nMpH: 7.5Assay Description:N-terminally His-tagged PI3K alpha (Cat. No. PV4789; 0.49 mg/ml), Alexa Fluor 647 labeled kinase Tracer 314 (Cat. No. PV6087), Biotin anti-His Tag an...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM228152((R)-5-(4-morpholino-5a,6,8,9-tetrahydro-5H- pyrimi...)
Affinity DataKi:  42nM IC50: 411nMpH: 7.5Assay Description:N-terminally His-tagged PI3K alpha (Cat. No. PV4789; 0.49 mg/ml), Alexa Fluor 647 labeled kinase Tracer 314 (Cat. No. PV6087), Biotin anti-His Tag an...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM228158((S)-5-(2-morpholino-5a,6,8,9-tetrahydro-5H- pyrimi...)
Affinity DataKi:  166nM IC50: 1.64E+3nMpH: 7.5Assay Description:N-terminally His-tagged PI3K alpha (Cat. No. PV4789; 0.49 mg/ml), Alexa Fluor 647 labeled kinase Tracer 314 (Cat. No. PV6087), Biotin anti-His Tag an...More data for this Ligand-Target Pair
In DepthDetails
US Patent