Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 8545
TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212270(US9504684, Ex.-1 | 6-(6-amino-5-methylpyrazin-2-yl...)
Affinity DataIC50: 6.20nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212276(US9504684, Ex.-7 | 2-(5-((6-(6-amino-5-methylpyraz...)
Affinity DataIC50: 8.70nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212274(US9504684, Ex.-5 | 2-(5-((6-(6-aminopyrazin-2-yl)i...)
Affinity DataIC50: 12.2nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212272(US9504684, Ex.-3 | (R)-(4-(4-((6-(6-aminopyrazin-2...)
Affinity DataIC50: 13.3nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212271(US9504684, Ex.-2 | 6-(6-aminopyrazin-2-yl)-N-(4-(4...)
Affinity DataIC50: 13.5nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212275(US9504684, Ex.-6 | 2-((4-(4-((6-(6-aminopyrazin-2-...)
Affinity DataIC50: 14.5nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212279(US9504684, 6-(5-amino-6-methylpyridin-3-yl)-N-(4-m...)
Affinity DataIC50: 16nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212277(US9504684, 6-(5-aminopyridin-3-yl)-N-(4-morpholino...)
Affinity DataIC50: 31nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212273(US9504684, Ex.-4 | 6-(6-aminopyrazin-2-yl)-5-methy...)
Affinity DataIC50: 44nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212280(US9504684, 6-(6-aminopyridin-3-yl)-N-(3,4-dimethox...)
Affinity DataIC50: 53nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTyrosine-protein kinase SYK(Human)
Gilead Sciences

US Patent
LigandPNGBDBM212278(US9504684, 6-(3-aminophenyl)-N-(3,4-dimethoxypheny...)
Affinity DataIC50: 188nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails
US Patent