Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 8353
TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242688(US9422290, I-1)
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242702(US9422290, II-9)
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242714(US9422290, III-3)
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242696(US9422290, II-3)
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242713(US9422290, III-2)
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242701(US9422290, II-8)
Affinity DataIC50: 4nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242700(US9422290, II-7)
Affinity DataIC50: 8nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242699(US9422290, II-6)
Affinity DataIC50: 8nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242694(US9422290, II-1)
Affinity DataIC50: 10nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242691(US9422290, I-4)
Affinity DataIC50: 25nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242704(US9422290, II-14)
Affinity DataIC50: 26nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242705(US9422290, II-15)
Affinity DataIC50: 29nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242708(US9422290, II-18)
Affinity DataIC50: 31nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242687(US9422290, III-8 | US9422290, III-6)
Affinity DataIC50: 32nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242687(US9422290, III-8 | US9422290, III-6)
Affinity DataIC50: 33nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242697(US9422290, II-4)
Affinity DataIC50: 37nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242686(US9422290, III-7 | US9422290, III-5)
Affinity DataIC50: 37nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242703(US9422290, II-10)
Affinity DataIC50: 38nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242720(US9422290, III-11)
Affinity DataIC50: 39nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242718(US9422290, III-9)
Affinity DataIC50: 40nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242715(US9422290, III-4)
Affinity DataIC50: 40nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242710(US9422290, II-20)
Affinity DataIC50: 43nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242719(US9422290, III-10)
Affinity DataIC50: 44nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242684(US9422290, II-12)
Affinity DataIC50: 51nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242686(US9422290, III-7 | US9422290, III-5)
Affinity DataIC50: 57nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242712(US9422290, III-1)
Affinity DataIC50: 61nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242683(US9422290, II-11)
Affinity DataIC50: 64nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242690(US9422290, I-3)
Affinity DataIC50: 67nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242711(US9422290, II-21)
Affinity DataIC50: 72nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242693(US9422290, I-6)
Affinity DataIC50: 74nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242689(US9422290, I-2)
Affinity DataIC50: 83nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242692(US9422290, I-5)
Affinity DataIC50: 83nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242698(US9422290, II-5)
Affinity DataIC50: 105nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242709(US9422290, II-19)
Affinity DataIC50: 105nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242695(US9422290, II-2)
Affinity DataIC50: 117nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242707(US9422290, II-17)
Affinity DataIC50: 140nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242706(US9422290, II-16)
Affinity DataIC50: 711nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM242685(US9422290, II-13)
Affinity DataIC50: 2.00E+3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
Go to US Patent