Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 8079
TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232961(US9353113, 10(5))
Affinity DataIC50: 3.80nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
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Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232952(US9353113, 3(50) | US9862721, 3(50))
Affinity DataIC50: 4.5nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
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Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232957(US9353113, 7(41) | US9862721, 7(41))
Affinity DataIC50: 4.90nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
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Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232955(US9353113, 6(65) | US9862721, 6(65))
Affinity DataIC50: 5.10nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
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Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232962(US9353113, 11(12) | US9862721, 11(12))
Affinity DataIC50: 5.40nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
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Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232954(US9353113, 6(63) | US9862721, 6(63))
Affinity DataIC50: 8nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
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Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232963(US9353113, 11(24) | US9862721, 11(24))
Affinity DataIC50: 8.40nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232953(US9353113, 6(53) | US9862721, 6(53))
Affinity DataIC50: 10nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232959(US9353113, 9(1) | US9862721, 9(1))
Affinity DataIC50: 12nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
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Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232964(US9353113, Ref. Ex. 2)
Affinity DataIC50: 14nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
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Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232958(US9353113, 7(45) | US9862721, 7(45))
Affinity DataIC50: 16nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
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Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232960(US9353113, 10(2))
Affinity DataIC50: 17nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details
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TargetAutotaxin(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM232956(US9353113, 7(3) | US9862721, 7(3))
Affinity DataIC50: 28nMpH: 9.0Assay Description:10 μL of a test compound solution (10% dimethyl sulfoxide) at each concentration and 40 μL of a 5 μg/mL human ENPP2 solution (buffer A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details
Go to US Patent