Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 7689
Target5-hydroxytryptamine receptor 1A/2C(Human)
Columbia University

US Patent
LigandPNGBDBM50024605(US9290463, E | CHEMBL3330603)
Affinity DataKi:  0.150nM ΔG°:  -52.1kJ/molepH: 7.4 T: 2°CAssay Description:Preparation of Membrane Fractions from CHO-h5-HT1A Cells. Membranes from CHO cells stably expressing the human 5-HT1A receptor at a density of 8 pmol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2017
Entry Details
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Target5-hydroxytryptamine receptor 1A/2C(Human)
Columbia University

US Patent
LigandPNGBDBM50024573(US9290463, A | CHEMBL3330617)
Affinity DataKi:  4nM ΔG°:  -44.6kJ/molepH: 7.4 T: 2°CAssay Description:Preparation of Membrane Fractions from CHO-h5-HT1A Cells. Membranes from CHO cells stably expressing the human 5-HT1A receptor at a density of 8 pmol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2017
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 1A/2C(Human)
Columbia University

US Patent
LigandPNGBDBM210829(US9290463, B)
Affinity DataKi:  5.5nM ΔG°:  -43.8kJ/molepH: 7.4 T: 2°CAssay Description:Preparation of Membrane Fractions from CHO-h5-HT1A Cells. Membranes from CHO cells stably expressing the human 5-HT1A receptor at a density of 8 pmol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2017
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 1A/2C(Human)
Columbia University

US Patent
LigandPNGBDBM210830(US9290463, D)
Affinity DataKi:  6nM ΔG°:  -43.6kJ/molepH: 7.4 T: 2°CAssay Description:Preparation of Membrane Fractions from CHO-h5-HT1A Cells. Membranes from CHO cells stably expressing the human 5-HT1A receptor at a density of 8 pmol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2017
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 1A/2C(Human)
Columbia University

US Patent
LigandPNGBDBM50024603(US9290463, C | CHEMBL3330604)
Affinity DataKi:  58.3nM ΔG°:  -38.4kJ/molepH: 7.4 T: 2°CAssay Description:Preparation of Membrane Fractions from CHO-h5-HT1A Cells. Membranes from CHO cells stably expressing the human 5-HT1A receptor at a density of 8 pmol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2017
Entry Details
Go to US Patent