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Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 7431
TargetCoagulation factor X(Human)
Portola Pharmaceuticals

US Patent
LigandPNGBDBM194506(US9200268, Table 4, Compound 2)
Affinity DataIC50: 24nMpH: 7.4 T: 2°CAssay Description:All assays, which are performed in 96-well microtiter plates, measure proteolytic activity of the enzyme (factor Xa) by following cleavage of a paran...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2016
Entry Details
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TargetCoagulation factor X(Human)
Portola Pharmaceuticals

US Patent
LigandPNGBDBM194508(US9200268, Table 4, Compound 4)
Affinity DataIC50: 158nMpH: 7.4 T: 2°CAssay Description:All assays, which are performed in 96-well microtiter plates, measure proteolytic activity of the enzyme (factor Xa) by following cleavage of a paran...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2016
Entry Details
Go to US Patent

TargetCoagulation factor X(Human)
Portola Pharmaceuticals

US Patent
LigandPNGBDBM194505(US9200268, Table 4, Compound 1)
Affinity DataIC50: 227nMpH: 7.4 T: 2°CAssay Description:All assays, which are performed in 96-well microtiter plates, measure proteolytic activity of the enzyme (factor Xa) by following cleavage of a paran...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2016
Entry Details
Go to US Patent

TargetCoagulation factor X(Human)
Portola Pharmaceuticals

US Patent
LigandPNGBDBM194509(US9200268, Table 4, Compound 5)
Affinity DataIC50: 320nMpH: 7.4 T: 2°CAssay Description:All assays, which are performed in 96-well microtiter plates, measure proteolytic activity of the enzyme (factor Xa) by following cleavage of a paran...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2016
Entry Details
Go to US Patent

TargetCoagulation factor X(Human)
Portola Pharmaceuticals

US Patent
LigandPNGBDBM194507(US9200268, Table 4, Compound 3)
Affinity DataIC50: 615nMpH: 7.4 T: 2°CAssay Description:All assays, which are performed in 96-well microtiter plates, measure proteolytic activity of the enzyme (factor Xa) by following cleavage of a paran...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2016
Entry Details
Go to US Patent