Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 7387
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192505(US9187477, 1)
Affinity DataEC50:  1.20nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192506(US9187477, 2)
Affinity DataEC50:  32nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192507(US9187477, 3)
Affinity DataEC50:  108nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192508(US9187477, 16 | US9187477, 4)
Affinity DataEC50:  12nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192509(US9187477, 5)
Affinity DataEC50:  119nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192510(US9187477, 6)
Affinity DataEC50:  6nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192511(US9187477, 7)
Affinity DataEC50:  468nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192512(US9187477, 8)
Affinity DataEC50:  339nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192513(US9187477, 9)
Affinity DataEC50:  17nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192514(US9187477, 10)
Affinity DataEC50:  26nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192515(US9187477, 11)
Affinity DataEC50:  35nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192516(US9187477, 12)
Affinity DataEC50:  1.31E+3nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192517(US9187477, 13)
Affinity DataEC50:  2.04E+3nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192518(US9187477, 14)
Affinity DataEC50:  578nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192519(US9187477, 15)
Affinity DataEC50:  133nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM192508(US9187477, 16 | US9187477, 4)
Affinity DataEC50:  290nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In DepthDetails
US Patent