Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 7385
TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM192498(US9187470, 89)
Affinity DataIC50: 27.5nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM50249406(1-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-3-(4-(py...)
Affinity DataIC50: 82.7nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent
PDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM192497(US9187470, 62)
Affinity DataIC50: 281nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM50249406(1-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-3-(4-(py...)
Affinity DataIC50: 620nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent
PDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 1.97E+3nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM50303597((S)-2-(2-amino-3-phenylpropylamino)-3-methyl-5-(na...)
Affinity DataIC50: 7.74E+3nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM192500(US9187470, 115)
Affinity DataIC50: 8.65E+3nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM192499(US9187470, 117)
Affinity DataIC50: 1.02E+4nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM192502(US9187470, 124)
Affinity DataIC50: 1.49E+4nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent
PDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM192499(US9187470, 117)
Affinity DataIC50: 1.58E+4nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM192502(US9187470, 124)
Affinity DataIC50: 9.87E+4nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent
PDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 13(Human)
Washington University

US Patent
LigandPNGBDBM192501(US9187470, 104 (SB203580) | US10865384, Compound S...)
Affinity DataIC50: 8.76E+7nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
In DepthDetails
US Patent