Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 7279
TargetVascular endothelial growth factor receptor 2(Human)
Beta Pharma

US Patent
LigandPNGBDBM186015(US9163010, Formula II)
Affinity DataIC50: 2.5nMAssay Description:The effects of compound of formula II on inhibiting VEGFR were compared against that of sunitinib in vitro.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2016
Entry Details
Go to US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Beta Pharma

US Patent
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 10nMAssay Description:The effects of compound of formula II on inhibiting VEGFR were compared against that of sunitinib in vitro.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2016
Entry Details
Go to US Patent

TargetVascular endothelial growth factor receptor 1(Human)
Beta Pharma

US Patent
LigandPNGBDBM186015(US9163010, Formula II)
Affinity DataIC50: 40nMAssay Description:The effects of compound of formula II on inhibiting VEGFR were compared against that of sunitinib in vitro.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2016
Entry Details
Go to US Patent