Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 7218
TargetHistamine H4 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM60636(US9138431, S-NORKETOTIFEN (SNORK))
Affinity DataIC50: 1.10E+3nMAssay Description:Histamine H-4 Receptor Binding AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
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TargetHistamine H4 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM181150(US9333199, RS-NORKETOTIFEN (NORK) | US9138431, RS-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Histamine H-4 Receptor Binding AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
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TargetHistamine H4 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM60637(US9138431, R-NORKETOTIFEN (SNORK))
Affinity DataIC50: 2.30E+3nMAssay Description:Histamine H-4 Receptor Binding AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
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TargetHistamine H1 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM94597((Z)-2-butenedioate;10-(1-methyl-4-piperidinylidene...)
Affinity DataIC50: 2.30E+3nMAssay Description:Affinities of the test compounds for peripheral human histamine H-1-receptors were assessed using receptor-binding assays. The specific binding of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
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TargetHistamine H4 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM50017674(Hydramine | Benylin | Silphen | (2-Benzhydryloxy-e...)
Affinity DataIC50: 1.10E+4nMAssay Description:Histamine H-4 Receptor Binding AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
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TargetHistamine H1 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM181150(US9333199, RS-NORKETOTIFEN (NORK) | US9138431, RS-...)
Affinity DataIC50: 1.10E+4nMAssay Description:Affinities of the test compounds for peripheral human histamine H-1-receptors were assessed using receptor-binding assays. The specific binding of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
Go to US Patent

TargetHistamine H4 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM50073179(CHEMBL1172 | Clarinex | Claritin-D | Claritin | SC...)
Affinity DataIC50: 1.60E+4nMAssay Description:Histamine H-4 Receptor Binding AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
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TargetHistamine H1 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM50073179(CHEMBL1172 | Clarinex | Claritin-D | Claritin | SC...)
Affinity DataIC50: 1.60E+4nMAssay Description:Affinities of the test compounds for peripheral human histamine H-1-receptors were assessed using receptor-binding assays. The specific binding of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
Go to US Patent

TargetHistamine H1 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM60637(US9138431, R-NORKETOTIFEN (SNORK))
Affinity DataIC50: 1.70E+4nMAssay Description:Affinities of the test compounds for peripheral human histamine H-1-receptors were assessed using receptor-binding assays. The specific binding of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
Go to US Patent

TargetHistamine H4 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM94597((Z)-2-butenedioate;10-(1-methyl-4-piperidinylidene...)
Affinity DataIC50: 2.10E+4nMAssay Description:Histamine H-4 Receptor Binding AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
Go to US Patent

TargetHistamine H1 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM60636(US9138431, S-NORKETOTIFEN (SNORK))
Affinity DataIC50: 2.30E+4nMAssay Description:Affinities of the test compounds for peripheral human histamine H-1-receptors were assessed using receptor-binding assays. The specific binding of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
Go to US Patent

TargetHistamine H1 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM50017674(Hydramine | Benylin | Silphen | (2-Benzhydryloxy-e...)
Affinity DataIC50: 8.40E+4nMAssay Description:Affinities of the test compounds for peripheral human histamine H-1-receptors were assessed using receptor-binding assays. The specific binding of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
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TargetHistamine H1 receptor(Human)
Bridge Pharma

US Patent
LigandPNGBDBM22876(Sch 29851 | Claritin | CHEMBL998 | ethyl 4-{13-chl...)
Affinity DataIC50: 1.50E+6nMAssay Description:Affinities of the test compounds for peripheral human histamine H-1-receptors were assessed using receptor-binding assays. The specific binding of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2016
Entry Details
Go to US Patent