Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 7097
TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173858(US9102599, 2)
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173867(US9102599, 50)
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173866(US9102599, 47)
Affinity DataIC50: 14nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173864(US9102599, 44)
Affinity DataIC50: 19nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173868(US9102599, 53)
Affinity DataIC50: 25nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173860(US9102599, 6)
Affinity DataIC50: 30nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173871(US9102599, 122)
Affinity DataIC50: 129nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173862(US9102599, 27)
Affinity DataIC50: 132nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173863(US9102599, 43)
Affinity DataIC50: 134nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173869(US9102599, 94)
Affinity DataIC50: 184nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173870(US9102599, 112)
Affinity DataIC50: 248nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173872(US9102599, 133)
Affinity DataIC50: 1.09E+3nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173861(US9102599, 11)
Affinity DataIC50: 1.43E+3nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173865(US9102599, 45)
Affinity DataIC50: 2.81E+3nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCholesteryl ester transfer protein(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM173859(US9102599, 5)
Affinity DataIC50: 4.36E+3nMpH: 7.4 T: 2°CAssay Description:Compounds of the present invention inhibit CETP-dependent cholesterol ester transfer from HDL to LDL as described here. Dilutions of compounds in DMS...More data for this Ligand-Target Pair
In DepthDetails
US Patent