Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 6763
TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331713(5,7-dichloro-3-(trifluoromethyl)-1,2,3,4-tetrahydr...)
Affinity DataIC50: 13nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151588(US8987319, 9b)
Affinity DataIC50: 13nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331698(5,6-dichloro-9H-carbazol-1-ol | CHEMBL1288959)
Affinity DataIC50: 15nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151589(US8987319, 10)
Affinity DataIC50: 20nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151593(US8987319, 16)
Affinity DataIC50: 20nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331710(6,7-dichloro-1-(perfluoroethyl)-2,3,4,9-tetrahydro...)
Affinity DataIC50: 34nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331697(2-bromo-6,7-dichloro-9H-carbazol-1-ol | CHEMBL1288...)
Affinity DataIC50: 34nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331701(6,8-dichloro-1-(trifluoromethyl)-2,3,4,9-tetrahydr...)
Affinity DataIC50: 34nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151602(US8987319, 28)
Affinity DataIC50: 54nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151592(US8987319, 15)
Affinity DataIC50: 70nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331702(5,8-dichloro-1-(trifluoromethyl)-2,3,4,9-tetrahydr...)
Affinity DataIC50: 85nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331704(8-chloro-6-fluoro-1-(trifluoromethyl)-2,3,4,9-tetr...)
Affinity DataIC50: 90nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331712(6,8-dichloro-2,2-difluoro-1-(trifluoromethyl)-2,3,...)
Affinity DataIC50: 100nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151601(US8987319, 27)
Affinity DataIC50: 120nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151599(US8987319, 25)
Affinity DataIC50: 130nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151590(US8987319, 12)
Affinity DataIC50: 140nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151603(US8987319, 29)
Affinity DataIC50: 175nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151595(US8987319, 19)
Affinity DataIC50: 220nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151604(US8987319, 30)
Affinity DataIC50: 390nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151597(US8987319, 23)
Affinity DataIC50: 400nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151598(US8987319, 24)
Affinity DataIC50: 410nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331707(1-hydroxy-1-(trifluoromethyl)-2,3,4,9-tetrahydro-1...)
Affinity DataIC50: 480nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151591(US8987319, 14)
Affinity DataIC50: 520nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331703(2,4-dichloro-6-(trifluoromethyl)-5,6,7,8,9,10-hexa...)
Affinity DataIC50: 600nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151600(US8987319, 26)
Affinity DataIC50: 1.00E+3nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331699(2-benzyl-6,7-dichloro-9H-carbazol-1-ol | CHEMBL129...)
Affinity DataIC50: 1.00E+3nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151587(US8987319, 9a)
Affinity DataIC50: 1.00E+3nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331700(2-benzyl-5,6-dichloro-9H-carbazol-1-ol | CHEMBL129...)
Affinity DataIC50: 1.00E+3nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331695(6-bromo-9H-carbazol-1-ol | CHEMBL1288956)
Affinity DataIC50: 1.42E+3nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331708(6,7-dichloro-1-(trifluoromethyl)-2,3,4,9-tetrahydr...)
Affinity DataIC50: 1.56E+3nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331696(8-hydroxy-9H-carbazole-3-carbonitrile | CHEMBL1288...)
Affinity DataIC50: 4.60E+3nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331706(1-hydroxy-1-methyl-2,3,4,9-tetrahydro-1H-carbazole...)
Affinity DataIC50: 9.20E+3nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151596(US8987319, 21)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM151594(US8987319, 18)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331711(1-hydroxy-1-(perfluoroethyl)-2,3,4,9-tetrahydro-1H...)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331705(6,7-dichloro-1-methyl-2,3,4,9-tetrahydro-1H-carbaz...)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331709(5,6-dichloro-1-(trifluoromethyl)-2,3,4,9-tetrahydr...)
Affinity DataIC50: 4.02E+4nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In DepthDetails
US Patent