Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 6416
LigandPNGBDBM127925(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 0.180nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127929(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 0.290nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM127920(US8796304, 2-[2-(5,8-Bis(trideuteromethyl)-[1,2,4]...)
Affinity DataIC50: 0.400nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127920(US8796304, 2-[2-(5,8-Bis(trideuteromethyl)-[1,2,4]...)
Affinity DataIC50: 0.400nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127936(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 0.440nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127934(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 0.440nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127921(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 0.690nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127932(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 0.790nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127926(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 0.810nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127931(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 1.20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM127927(US8796304, 2-[2-(5,8-Dimethyl-7-oxy-[1,2,4]triazol...)
Affinity DataIC50: 2.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127928(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 3.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127923(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 4.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127922(US8796304, 2-[2-(5-Methyl-[1,2,4]triazolo[1,5-a]py...)
Affinity DataIC50: 6.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127933(US8796304, 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 6.90nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM127924(US8796304, {2-[2-(5H-Imidazo[2,1-a]isoindol-2-yl)-...)
Affinity DataIC50: 6.90nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127930(US8796304, 2-(2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1...)
Affinity DataIC50: 21nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM127938(US8796304, 2-[(5,7-dimethyl-[1,2,4]triazolo[1,5-a]...)
Affinity DataIC50: 260nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM127937(US8796304, 2-([1,2,4]Triazolo[1,5-a]pyridin-2-ylsu...)
Affinity DataIC50: 5.30E+3nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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US Patent