Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 6348
TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123905(US8754113, I-3-37)
Affinity DataIC50: 2nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123908(US8754113, I-3-56)
Affinity DataIC50: 4nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123898(US8754113, I-3-4)
Affinity DataIC50: 4nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123891(US8754113, I-1-85 | US9169240, 24)
Affinity DataIC50: 5nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123890(US8754113, I-1-83)
Affinity DataIC50: 6nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123907(US8754113, I-3-48)
Affinity DataIC50: 8nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123915(US8754113, A-10)
Affinity DataIC50: 8nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123913(US8754113, I-3-163)
Affinity DataIC50: 9nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123900(US8754113, I-3-11)
Affinity DataIC50: 9nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123914(US8754113, A-9)
Affinity DataIC50: 11nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123893(US8754113, I-2-197)
Affinity DataIC50: 12nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123922(US8754113, A-29)
Affinity DataIC50: 14nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123906(US8754113, I-3-41)
Affinity DataIC50: 14nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123894(US8754113, I-2-198)
Affinity DataIC50: 15nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123916(US8754113, A-13)
Affinity DataIC50: 22nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123912(US8754113, I-3-146)
Affinity DataIC50: 27nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123909(US8754113, I-3-93)
Affinity DataIC50: 28nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123892(US8754113, I-2-196)
Affinity DataIC50: 36nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123918(US8754113, A-17)
Affinity DataIC50: 41nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123921(US8754113, A-25)
Affinity DataIC50: 42nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123910(US8754113, I-3-112)
Affinity DataIC50: 44nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
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Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123904(US8754113, I-3-30)
Affinity DataIC50: 46nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123899(US8754113, I-3-6)
Affinity DataIC50: 52nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123889(US8754113, I-1-82)
Affinity DataIC50: 52nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123920(US8754113, A-21)
Affinity DataIC50: 65nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123911(US8754113, I-3-145)
Affinity DataIC50: 69nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123885(US8754113, I-1-23)
Affinity DataIC50: 73nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123901(US8754113, I-3-12)
Affinity DataIC50: 78nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123887(US8754113, I-1-31)
Affinity DataIC50: 83nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123886(US8754113, I-1-27)
Affinity DataIC50: 85nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123919(US8754113, A-19)
Affinity DataIC50: 110nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123917(US8754113, A-14)
Affinity DataIC50: 160nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123895(US8754113, I-2-204)
Affinity DataIC50: 190nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123902(US8754113, I-3-21)
Affinity DataIC50: 250nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123884(US8754113, I-1-9)
Affinity DataIC50: 260nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123888(US8754113, I-1-43)
Affinity DataIC50: 390nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123903(US8754113, I-3-23)
Affinity DataIC50: 400nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123896(US8754113, I-2-215)
Affinity DataIC50: 2.50E+3nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM123897(US8754113, I-2-216)
Affinity DataIC50: 2.30E+4nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
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