Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 6141
TargetTyrosine-protein kinase BTK(Human)
Roche Palo Alto

US Patent
LigandPNGBDBM111588(US8822457, II-3 | US8618098, II-3)
Affinity DataIC50: 18nMAssay Description:The assay is a capture of radioactive 33P phosphorylated product through filtration. The interactions of Btk, biotinylated SH2 peptide substrate (Src...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2014
Entry Details
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TargetTyrosine-protein kinase BTK(Human)
Roche Palo Alto

US Patent
LigandPNGBDBM111587(US8822457, II-1 | US8618098, II-1)
Affinity DataIC50: 22nMAssay Description:The assay is a capture of radioactive 33P phosphorylated product through filtration. The interactions of Btk, biotinylated SH2 peptide substrate (Src...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Roche Palo Alto

US Patent
LigandPNGBDBM111586(US8822457, I-1 | US8618098, I-1)
Affinity DataIC50: 112nMAssay Description:The assay is a capture of radioactive 33P phosphorylated product through filtration. The interactions of Btk, biotinylated SH2 peptide substrate (Src...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2014
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetTyrosine-protein kinase BTK(Human)
Roche Palo Alto

US Patent
LigandPNGBDBM111589(US8822457, III-1 | US8618098, III-1)
Affinity DataIC50: 124nMAssay Description:The assay is a capture of radioactive 33P phosphorylated product through filtration. The interactions of Btk, biotinylated SH2 peptide substrate (Src...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2014
Entry Details
Go to US Patent