Compile Data Set for Download or QSAR
Report error Found 302 Enz. Inhib. hit(s) with all data for entry = 6134
LigandPNGBDBM111368(US8614253, 32-4 | US9493435, 168 | US9241942, 32-4)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM111376(US8614253, 33-3 | US8614253, 32-12 | US9241942, 33...)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111376(US8614253, 33-3 | US8614253, 32-12 | US9241942, 33...)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111339(US8614253, 28-15 | US9241942, 28-13)
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111406(US8614253, 38-7 | US9241942, 38-7)
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111336(US8614253, 42-2 | US8614253, 28-12 | US9241942, 42...)
Affinity DataIC50: 19nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111336(US8614253, 42-2 | US8614253, 28-12 | US9241942, 42...)
Affinity DataIC50: 19nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111303(US8614253, 43-63 | US9241942, 27-63)
Affinity DataIC50: 21nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110983(US8614253, 43-5 | US8614253, 42-12 | US8614253, 3-...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110983(US8614253, 43-5 | US8614253, 42-12 | US8614253, 3-...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111342(US8614253, 29-2 | US9241942, 29-2)
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111405(US8614253, 38-6 | US9241942, 38-6)
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111358(US8614253, 29-18 | US9241942, 29-18)
Affinity DataIC50: 26nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110970(US8614253, 3-1 | US9241942, 3-1 | US9963434, Compo...)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110971(US8614253, 3-2 | US9241942, 3-2 | US9963434, Compo...)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111304(US8614253, 43-64 | US9241942, 27-64)
Affinity DataIC50: 32nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110972(US8614253, 43-10 | US8614253, 3-3 | US9241942, 3-3...)
Affinity DataIC50: 34nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111404(US8614253, 38-5 | US9241942, 38-5)
Affinity DataIC50: 34nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111346(US8614253, 42-4 | US8614253, 29-6 | US9241942, 42-...)
Affinity DataIC50: 36nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111346(US8614253, 42-4 | US8614253, 29-6 | US9241942, 42-...)
Affinity DataIC50: 36nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111247(US8614253, 43-7 | US9241942, 27-7)
Affinity DataIC50: 39nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110972(US8614253, 43-10 | US8614253, 3-3 | US9241942, 3-3...)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111335(US8614253, 28-11 | US9241942, 28-9)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111251(US8614253, 43-11 | US9241942, 27-11)
Affinity DataIC50: 42nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111383(US8614253, 42-9 | US8614253, 34-2 | US9241942, 42-...)
Affinity DataIC50: 45nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111383(US8614253, 42-9 | US8614253, 34-2 | US9241942, 42-...)
Affinity DataIC50: 45nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111234(US8614253, 26-21 | US9241942, 26-21)
Affinity DataIC50: 46nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111282(US8614253, 43-42 | US9241942, 27-42)
Affinity DataIC50: 46nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111370(US8614253, 32-6 | US9493435, 180 | US9241942, 32-6)
Affinity DataIC50: 47nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111420(US8614253, 40-1 | US9241942, 40-1)
Affinity DataIC50: 47nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111373(US8614253, 42-6 | US8614253, 32-9 | US9493435, 169...)
Affinity DataIC50: 48nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111373(US8614253, 42-6 | US8614253, 32-9 | US9493435, 169...)
Affinity DataIC50: 48nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111267(US8614253, 43-27 | US9241942, 27-27)
Affinity DataIC50: 61nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111334(US8614253, 28-10 | US9241942, 28-8)
Affinity DataIC50: 66nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111343(US8614253, 29-3 | US9241942, 29-3)
Affinity DataIC50: 66nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111372(US8614253, 32-8 | US9241942, 32-8)
Affinity DataIC50: 67nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110973(US8614253, 43-81 | US8614253, 3-4 | US9241942, 3-4...)
Affinity DataIC50: 70nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111228(US8614253, 26-15 | US9241942, 26-15)
Affinity DataIC50: 74nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111262(US8614253, 43-22 | US9241942, 27-22)
Affinity DataIC50: 74nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111344(US8614253, 29-4 | US9241942, 29-4)
Affinity DataIC50: 74nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110973(US8614253, 43-81 | US8614253, 3-4 | US9241942, 3-4...)
Affinity DataIC50: 79nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111345(US8614253, 29-5 | US9241942, 29-5)
Affinity DataIC50: 79nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110974(US8614253, 3-5 | US9241942, 3-5 | US9963434, Compo...)
Affinity DataIC50: 80nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM110975(US8614253, 43-4 | US8614253, 3-6 | US9241942, 3-6 ...)
Affinity DataIC50: 80nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111269(US8614253, 43-29 | US9241942, 27-29)
Affinity DataIC50: 81nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111230(US8614253, 26-17 | US9241942, 26-17)
Affinity DataIC50: 82nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111276(US8614253, 43-36 | US9241942, 27-36)
Affinity DataIC50: 82nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111331(US8614253, 28-7 | US9241942, 28-7)
Affinity DataIC50: 84nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111314(US8614253, 43-74 | US9241942, 27-74)
Affinity DataIC50: 85nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
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LigandPNGBDBM111271(US8614253, 43-31 | US9241942, 27-31)
Affinity DataIC50: 88nMpH: 7.5 T: 2°CAssay Description:IRE-1 alpha, T1 RNase, and RNase A assays carried out in vitro with several o-vanillin derivatives to demonstrate selectivity of the derivatives for ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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