Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 6101
TargetAdenosine receptor A1(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97464(US8609833, 17 | US8470800, A | US8609833, 86)
Affinity DataKi:  0.970nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A1(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97465(US8609833, 85 | US8470800, B)
Affinity DataKi:  2.63nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A1(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108258(US8609833, 91)
Affinity DataKi:  4.05nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A1(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108256(US8609833, 87 | CHEMBL2205239)
Affinity DataKi:  5.79nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A1(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108257(US8609833, 88)
Affinity DataKi:  7nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A1(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97467(US8609833, 93 | US8470800, D)
Affinity DataKi:  10.6nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A3(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108256(US8609833, 87 | CHEMBL2205239)
Affinity DataKi:  216nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A3(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97465(US8609833, 85 | US8470800, B)
Affinity DataKi:  513nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A3(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97464(US8609833, 17 | US8470800, A | US8609833, 86)
Affinity DataKi:  704nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A3(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108257(US8609833, 88)
Affinity DataKi:  900nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A2(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108256(US8609833, 87 | CHEMBL2205239)
Affinity DataKi:  951nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A3(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108258(US8609833, 91)
Affinity DataKi:  1.02E+3nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A3(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97467(US8609833, 93 | US8470800, D)
Affinity DataKi:  2.02E+3nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A2(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97465(US8609833, 85 | US8470800, B)
Affinity DataKi:  4.19E+3nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A2(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97464(US8609833, 17 | US8470800, A | US8609833, 86)
Affinity DataKi:  4.69E+3nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A2(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108258(US8609833, 91)
Affinity DataKi:  9.11E+3nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A2(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108257(US8609833, 88)
Affinity DataKi:  1.00E+4nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAdenosine receptor A2(Human)
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97467(US8609833, 93 | US8470800, D)
Affinity DataKi: >1.00E+5nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails
US Patent