Compile Data Set for Download or QSAR
Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 5974
Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103345(US8546392, 69)
Affinity DataIC50: 7nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103342(US8546392, 64)
Affinity DataIC50: 10nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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TargetCytochrome P450 1A2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103338(US8546392, 59)
Affinity DataIC50: 14nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103336(US8546392, 57)
Affinity DataIC50: 20nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103338(US8546392, 59)
Affinity DataIC50: 20nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335815(CHEMBL1650658 | US8546392, 72 | US8546392, 56 | N-...)
Affinity DataIC50: 23nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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TargetCytochrome P450 2C9(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103346(US8546392, 70)
Affinity DataIC50: 30nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103346(US8546392, 70)
Affinity DataIC50: 30nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335820(CHEMBL1650647 | US8546392, 68 | US8546392, 52 | 6-...)
Affinity DataIC50: 39nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103337(US8546392, 58)
Affinity DataIC50: 40nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103340(US8546392, 62)
Affinity DataIC50: 50nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103344(US8546392, 68)
Affinity DataIC50: 50nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103347(US8546392, 71)
Affinity DataIC50: 60nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103334(US8546392, 19)
Affinity DataIC50: 70nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103339(US8546392, 60)
Affinity DataIC50: 90nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103343(US8546392, 66)
Affinity DataIC50: 114nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103341(US8546392, 63)
Affinity DataIC50: 140nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 2C9(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103338(US8546392, 59)
Affinity DataIC50: 150nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103346(US8546392, 70)
Affinity DataIC50: 195nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103338(US8546392, 59)
Affinity DataIC50: 221nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
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TargetCytochrome P450 2C9(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335817(CHEMBL1650646 | US8546392, 70 | US8546392, 54 | 6-...)
Affinity DataIC50: 224nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 1A2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335817(CHEMBL1650646 | US8546392, 70 | US8546392, 54 | 6-...)
Affinity DataIC50: 259nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103342(US8546392, 64)
Affinity DataIC50: 403nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103340(US8546392, 62)
Affinity DataIC50: 458nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335817(CHEMBL1650646 | US8546392, 70 | US8546392, 54 | 6-...)
Affinity DataIC50: 500nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103335(US8546392, 42)
Affinity DataIC50: 500nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103337(US8546392, 58)
Affinity DataIC50: 527nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335815(CHEMBL1650658 | US8546392, 72 | US8546392, 56 | N-...)
Affinity DataIC50: 540nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335820(CHEMBL1650647 | US8546392, 68 | US8546392, 52 | 6-...)
Affinity DataIC50: 583nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103345(US8546392, 69)
Affinity DataIC50: 601nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 2C19(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335815(CHEMBL1650658 | US8546392, 72 | US8546392, 56 | N-...)
Affinity DataIC50: 680nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 1(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335817(CHEMBL1650646 | US8546392, 70 | US8546392, 54 | 6-...)
Affinity DataIC50: 840nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 2C19(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103338(US8546392, 59)
Affinity DataIC50: 880nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103336(US8546392, 57)
Affinity DataIC50: 959nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 2C9(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103334(US8546392, 19)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335815(CHEMBL1650658 | US8546392, 72 | US8546392, 56 | N-...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103338(US8546392, 59)
Affinity DataIC50: 1.16E+3nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 2C19(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335817(CHEMBL1650646 | US8546392, 70 | US8546392, 54 | 6-...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 2C9(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335815(CHEMBL1650658 | US8546392, 72 | US8546392, 56 | N-...)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103334(US8546392, 19)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103344(US8546392, 68)
Affinity DataIC50: 1.76E+3nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM50335817(CHEMBL1650646 | US8546392, 70 | US8546392, 54 | 6-...)
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103346(US8546392, 70)
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103339(US8546392, 60)
Affinity DataIC50: 2.94E+3nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 1A2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103334(US8546392, 19)
Affinity DataIC50: 3.99E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103335(US8546392, 42)
Affinity DataIC50: 4.19E+3nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 1A2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103338(US8546392, 59)
Affinity DataIC50: 5.34E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

Target17-beta-hydroxysteroid dehydrogenase type 2(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103334(US8546392, 19)
Affinity DataIC50: 5.64E+3nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 2C19(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103334(US8546392, 19)
Affinity DataIC50: 7.54E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

TargetCytochrome P450 2C19(Human)
Universitaet Des Saarlandes

US Patent
LigandPNGBDBM103346(US8546392, 70)
Affinity DataIC50: 8.83E+3nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2013
Entry Details
Go to US Patent

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