Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 5960
TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101030(US8507479, 674)
Affinity DataIC50: 10nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101029(US8507479, 669)
Affinity DataIC50: 10nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101023(US8507479, 655)
Affinity DataIC50: 10nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101026(US8507479, 664)
Affinity DataIC50: 20nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101032(US8507479, 689)
Affinity DataIC50: 40nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101031(US8507479, 680)
Affinity DataIC50: 50nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101022(US8507479, 652)
Affinity DataIC50: 60nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM2677(US8507479, 140 | US8541408, 80 | US8507479, 80)
Affinity DataIC50: 70nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100987(US8507479, 3)
Affinity DataIC50: 80nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101021(US8507479, 164)
Affinity DataIC50: 80nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101007(US8507479, 101)
Affinity DataIC50: 80nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101005(US8507479, 93)
Affinity DataIC50: 80nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101004(US8507479, 92)
Affinity DataIC50: 80nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100997(US8507479, 70)
Affinity DataIC50: 90nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101003(US8507479, 87)
Affinity DataIC50: 90nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101010(US8507479, 109)
Affinity DataIC50: 100nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100991(US8507479, 34)
Affinity DataIC50: 100nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100999(US8507479, 72)
Affinity DataIC50: 110nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101024(US8507479, 660)
Affinity DataIC50: 110nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101014(US8507479, 136)
Affinity DataIC50: 110nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101009(US8507479, 106)
Affinity DataIC50: 120nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101015(US8507479, 141)
Affinity DataIC50: 120nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101008(US8507479, 105)
Affinity DataIC50: 130nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100992(US8507479, 38)
Affinity DataIC50: 140nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100993(US8507479, 41)
Affinity DataIC50: 150nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100996(US8507479, 66)
Affinity DataIC50: 150nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101034(US8507479, 702)
Affinity DataIC50: 160nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101012(US8507479, 114)
Affinity DataIC50: 160nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100989(US8541408, 12 | US8507479, 12)
Affinity DataIC50: 160nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100998(US8507479, 71)
Affinity DataIC50: 160nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100988(US8541408, 11 | US8507479, 11)
Affinity DataIC50: 170nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101006(US8507479, 94)
Affinity DataIC50: 170nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101025(US8507479, 662)
Affinity DataIC50: 170nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100994(US8507479, 62)
Affinity DataIC50: 170nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101000(US8507479, 76)
Affinity DataIC50: 180nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101011(US8507479, 111)
Affinity DataIC50: 180nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101002(US8507479, 86)
Affinity DataIC50: 190nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101033(US8507479, 701)
Affinity DataIC50: 200nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101028(US8507479, 668)
Affinity DataIC50: 510nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM100995(US8507479, 65)
Affinity DataIC50: 720nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101027(US8507479, 665)
Affinity DataIC50: 870nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101013(US8507479, 126)
Affinity DataIC50: 2.14E+3nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101017(US8507479, 150)
Affinity DataIC50: 2.48E+3nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM102916(US8541408, 26)
Affinity DataIC50: 4.85E+3nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM9487(US8507479, 155 | US8541408, 155)
Affinity DataIC50: 5.96E+3nMAssay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101018(US8507479, 151)
Affinity DataIC50: 6.77E+3nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101020(US8507479, 163)
Affinity DataIC50: 6.79E+3nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM101016(US8507479, 149)
Affinity DataIC50: 9.25E+3nMpH: 7.0Assay Description:Inhibition assay using human BACE-1.More data for this Ligand-Target Pair
In DepthDetails
US Patent