Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 5922
TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100743(US8507714, 67)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100749(US8507714, 214)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100752(US8507714, 269)
Affinity DataIC50: 24nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100740(CHEMBL391608 | US8507714, 29)
Affinity DataIC50: 34nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100744(US8507714, 90)
Affinity DataIC50: 93nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100746(US8507714, 277 | US8507714, 150 | CHEMBL246560)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100739(US8507714, 15)
Affinity DataIC50: 160nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100746(US8507714, 277 | US8507714, 150 | CHEMBL246560)
Affinity DataIC50: 160nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100745(US8507714, 91)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100750(CHEMBL2397003 | US8507714, 239)
Affinity DataIC50: 260nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100742(US8507714, 61)
Affinity DataIC50: 260nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM2228(US8507714, 178A)
Affinity DataIC50: 300nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100747(CHEMBL2397007 | US8507714, 151)
Affinity DataIC50: 380nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100741(US8507714, 37)
Affinity DataIC50: 390nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100751(US8507714, 263)
Affinity DataIC50: 460nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM609(penicillin deriv. 23 | US8507714, 4)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100753(US8507714, 272)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM100754(US8507714, 285)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
Go to US Patent