Compile Data Set for Download or QSAR
Report error Found 99 Enz. Inhib. hit(s) with all data for entry = 12394
TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700357(US20240336593, Example 116 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700369(US20240336593, Example 130 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700368(US20240336593, Example 129 | Trans-(4-(3,4-dihydro...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700367(US20240336593, Example 128 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700366(US20240336593, Example 127 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700365(US20240336593, Example 124 | Preparation of 1-(4-(...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700364(US20240336593, Example 123 | Preparation of methyl...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700363(US20240336593, Example 122 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700362(US20240336593, Example 121 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700361(US20240336593, Example 120 | 1-(4-((6-(trans-4-(3,...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700360(US20240336593, Example 119 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700359(US20240336593, Example 118 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700358(US20240336593, Example 117 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700370(US20240336593, Example 131 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700356(US20240336593, Example 115 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700355(US20240336593, Example 113 | Preparation of 1-(4-(...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700354(US20240336593, Example 112 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700353(US20240336593, Example 111 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700352(US20240336593, Example 110 | Preparation of t-buty...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700351(US20240336593, Example 109 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700350(US20240336593, Example 108 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700349(US20240336593, Example 107 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700348(US20240336593, Example 106 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700347(US20240336593, Example 105 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700346(US20240336593, Example 104 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700382(US20240336593, Example 145)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700394(US20240336593, Example 157)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700393(US20240336593, Example 156)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700392(US20240336593, Example 155)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700391(US20240336593, Example 154)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700390(US20240336593, Example 153)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700389(US20240336593, Example 152)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700388(US20240336593, Example 151)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700387(US20240336593, Example 150)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700386(US20240336593, Example 149)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700385(US20240336593, Example 148)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700384(US20240336593, Example 147)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700383(US20240336593, Example 146)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700345(US20240336593, Example 103 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700381(US20240336593, Example 144)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700380(US20240336593, Example 143)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700379(US20240336593, Example 142)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700378(US20240336593, Example 141)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700377(US20240336593, Example 140)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700376(US20240336593, Example 139 | Preparation of 1-(4-(...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700375(US20240336593, Example 138 | Preparation of 4-((6-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700374(US20240336593, Example 135 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700373(US20240336593, Example 134 | Preparation of trans-...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700372(US20240336593, Example 133 | Preparation of (trans...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
lnnovStoneTherapeutics Limited

US Patent
LigandPNGBDBM700371(US20240336593, Example 132 | Preparation of (trans...)
Affinity DataIC50: 100nMAssay Description:Test method: A 1× enzyme reaction buffer (10 mM Tris 8.0 (Sigma, Cat. No. T2694-1L), 0.01% Tween-20 (Sigma, Cat. No. P2287-100 ML), 1 mM DTT (Sigma, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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