Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 12249
TargetSigma non-opioid intracellular receptor 1(Human)
Prilenia Neurotherapeutics

US Patent
LigandPNGBDBM50308028(4-[3-(Methylsulfonyl)phenyl]-1-propylpiperidine | ...)
Affinity DataKi:  57nMAssay Description:In vitro binding assay performed at Eurofins Panlabs Taiwan, ltd. Specific ligand binding was determined in the presence of an excess of unlabelled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2024
Entry Details
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TargetSigma non-opioid intracellular receptor 1(Human)
Prilenia Neurotherapeutics

US Patent
LigandPNGBDBM638725(US20230390272, Compound 1 | US20240261273, Compoun...)
Affinity DataKi:  370nMAssay Description:In vitro binding assay performed at Eurofins Panlabs Taiwan, ltd. Specific ligand binding was determined in the presence of an excess of unlabelled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2024
Entry Details
Go to US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
Prilenia Neurotherapeutics

US Patent
LigandPNGBDBM638726(US20230390272, Compound 4 | US20240261273, Compoun...)
Affinity DataKi:  2.90E+3nMAssay Description:In vitro binding assay performed at Eurofins Panlabs Taiwan, ltd. Specific ligand binding was determined in the presence of an excess of unlabelled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2024
Entry Details
Go to US Patent

TargetSigma intracellular receptor 2(Human)
Prilenia Neurotherapeutics

US Patent
LigandPNGBDBM50308028(4-[3-(Methylsulfonyl)phenyl]-1-propylpiperidine | ...)
Affinity DataKi:  5.45E+3nMAssay Description:In vitro binding assay performed at Eurofins Panlabs Taiwan, ltd. Specific ligand binding was determined in the presence of an excess of unlabelled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2024
Entry Details
Go to US Patent

TargetSigma intracellular receptor 2(Human)
Prilenia Neurotherapeutics

US Patent
LigandPNGBDBM638725(US20230390272, Compound 1 | US20240261273, Compoun...)
Affinity DataKi: >1.00E+5nMAssay Description:In vitro binding assay performed at Eurofins Panlabs Taiwan, ltd. Specific ligand binding was determined in the presence of an excess of unlabelled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2024
Entry Details
Go to US Patent

TargetSigma intracellular receptor 2(Human)
Prilenia Neurotherapeutics

US Patent
LigandPNGBDBM638726(US20230390272, Compound 4 | US20240261273, Compoun...)
Affinity DataKi: >1.00E+5nMAssay Description:In vitro binding assay performed at Eurofins Panlabs Taiwan, ltd. Specific ligand binding was determined in the presence of an excess of unlabelled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2024
Entry Details
Go to US Patent