Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 12073
Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676496(US20240166639, Example 41)
Affinity DataKi:  0.300nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676494(US20240166639, Example 39)
Affinity DataKi:  0.400nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676503(4-bromo-3-(2-(dimethylamino)ethoxy)-N-(6-(2-fluoro...)
Affinity DataKi:  0.5nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM85166(CAS_3292447 | NSC_3292447 | SB 216641 | US20240166...)
Affinity DataKi:  0.600nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676498(US20240166639, Example 43)
Affinity DataKi:  1.5nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676497(US20240166639, Example 42)
Affinity DataKi:  2nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676495(US20240166639, Example 40)
Affinity DataKi:  3.5nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM50084959(4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)pheny...)
Affinity DataKi:  5.92nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676491(US20240166639, Example 21)
Affinity DataKi:  6.30nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM29644(APOMORPHINE HYDROCHLORIDE | SMR000059235 | APOMORP...)
Affinity DataKi:  6.92nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676492(US20240166639, Example 23)
Affinity DataKi:  7.90nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM50084959(4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)pheny...)
Affinity DataKi:  8.20nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676490(US20240166639, Example 7)
Affinity DataKi:  9.70nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676500(US20240166639, Example 47)
Affinity DataKi:  9.70nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676493(US20240166639, Example 38)
Affinity DataKi:  16.5nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676499(US20240166639, Example 45)
Affinity DataKi:  25.9nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676502(US20240166639, Example 54)
Affinity DataKi:  48.3nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM676501(US20240166639, Example 49)
Affinity DataKi:  126nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM85166(CAS_3292447 | NSC_3292447 | SB 216641 | US20240166...)
Affinity DataKi:  143nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676496(US20240166639, Example 41)
Affinity DataKi:  1.00E+3nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676503(4-bromo-3-(2-(dimethylamino)ethoxy)-N-(6-(2-fluoro...)
Affinity DataKi:  1.00E+3nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676495(US20240166639, Example 40)
Affinity DataKi:  1.50E+3nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 1B(Human)
Leukos Biotech

US Patent
LigandPNGBDBM29644(APOMORPHINE HYDROCHLORIDE | SMR000059235 | APOMORP...)
Affinity DataKi:  1.76E+3nMAssay Description:Serotonin 5-HT1B receptor competition binding experiments were carried out in a polypropylene 96-well plate. In each well was incubated 5 μg of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
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Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676498(US20240166639, Example 43)
Affinity DataKi:  2.00E+3nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676494(US20240166639, Example 39)
Affinity DataKi:  2.50E+3nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676490(US20240166639, Example 7)
Affinity DataKi:  2.50E+3nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676492(US20240166639, Example 23)
Affinity DataKi:  3.00E+3nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676497(US20240166639, Example 42)
Affinity DataKi:  3.50E+3nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676491(US20240166639, Example 21)
Affinity DataKi:  3.50E+3nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676501(US20240166639, Example 49)
Affinity DataKi: >1.00E+4nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676502(US20240166639, Example 54)
Affinity DataKi: >1.00E+4nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676500(US20240166639, Example 47)
Affinity DataKi: >1.00E+4nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676499(US20240166639, Example 45)
Affinity DataKi: >1.00E+4nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2A(Rat)
Leukos Biotech

US Patent
LigandPNGBDBM676493(US20240166639, Example 38)
Affinity DataKi: >1.00E+4nMAssay Description:Serotonin 5-HT2A receptor competition binding experiments were carried out in a polypropilene 96-well plate. In each well was incubated 80 μg of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
Go to US Patent