Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 11522
LigandPNGBDBM622599(US20230312601, Example 30)
Affinity DataEC50:  82nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622590(US20230312601, Example 21)
Affinity DataEC50:  141nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622591(US20230312601, Example 22)
Affinity DataEC50:  228nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622592(US20230312601, Example 23)
Affinity DataEC50:  139nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622593(US20230312601, Example 24)
Affinity DataEC50:  979nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622594(US20230312601, Example 25)
Affinity DataEC50:  67nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622595(US20230312601, Example 26)
Affinity DataEC50:  393nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622596(US20230312601, Example 27)
Affinity DataEC50:  70nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622597(US20230312601, Example 28)
Affinity DataEC50:  138nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622598(US20230312601, Example 29)
Affinity DataEC50:  232nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622589(US20230312601, Example 20)
Affinity DataEC50:  120nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622600(US20230312601, Example 31)
Affinity DataEC50:  82nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622601(US20230312601, Example 32)
Affinity DataEC50:  113nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622602(US20230312601, Example 33)
Affinity DataEC50:  162nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622603(US20230312601, Example 34)
Affinity DataEC50:  112nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622604(US20230312601, Example 35)
Affinity DataEC50:  500nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622605(US20230312601, Example 36)
Affinity DataEC50:  48nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622606(US20230312601, Example 37)
Affinity DataEC50:  60nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622607(US20230312601, Example 38)
Affinity DataEC50:  156nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622608(US20230312601, Example 39)
Affinity DataEC50:  83nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622580(US20230312601, Example 11)
Affinity DataEC50:  155nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622571(US20230312601, Example 2)
Affinity DataEC50:  190nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622572(US20230312601, Example 3)
Affinity DataEC50:  110nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622573(US20230312601, Example 4)
Affinity DataEC50:  158nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622574(US20230312601, Example 5)
Affinity DataEC50:  77nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622575(US20230312601, Example 6)
Affinity DataEC50:  146nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622576(US20230312601, Example 7)
Affinity DataEC50:  135nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622577(US20230312601, Example 8)
Affinity DataEC50:  99nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622578(US20230312601, Example 9)
Affinity DataEC50:  102nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622579(US20230312601, Example 10)
Affinity DataEC50:  198nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622570(US20230312601, Example 1)
Affinity DataEC50:  91nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622581(US20230312601, Example 12)
Affinity DataEC50:  61nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622582(US20230312601, Example 13)
Affinity DataEC50:  193nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622583(US20230312601, Example 14)
Affinity DataEC50:  97nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622584(US20230312601, Example 15)
Affinity DataEC50:  103nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622585(US20230312601, Example 16)
Affinity DataEC50:  106nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622586(US20230312601, Example 17)
Affinity DataEC50:  92nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622587(US20230312601, Example 18)
Affinity DataEC50:  284nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
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LigandPNGBDBM622588(US20230312601, Example 19)
Affinity DataEC50:  198nMAssay Description:A Quenched Fluorescence Resonance Energy Transfer (Quench-FRET) enzyme assay was used to test the ability of exemplary MALT-1 inhibitors Example 1 to...More data for this Ligand-Target Pair
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Date in BDB:
11/13/2023
Entry Details
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