Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 12627
TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716161(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(4-methyl-3- ...)
Affinity DataIC50: 0.130nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716154(6-(((1S,2S,4S)-4-(3-chloro-5- (trifluoromethyl)phe...)
Affinity DataIC50: 0.188nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716155(6-(((1S,2S,4S)-4-(3,5- dichlorophenyl)-2-(dimethyl...)
Affinity DataIC50: 0.222nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716141(6-(((1S,2S,4S)-4-(4-chloro-3- (trifluoromethyl)phe...)
Affinity DataIC50: 0.247nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716153(6-(((1S,2S,4S)-2-(ethyl- (methyl)amino)-4-(3- (tri...)
Affinity DataIC50: 0.272nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716124(5-chloro-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2-(1-...)
Affinity DataIC50: 0.281nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716142(6-(((1S,2S,4S)-4-(3,4-dichloro- phenyl)-2-(dimethy...)
Affinity DataIC50: 0.301nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716163(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(3-methyl-5- ...)
Affinity DataIC50: 0.351nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716123(5-chloro-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2-pyr...)
Affinity DataIC50: 0.388nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716159(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(2-methyl-5- ...)
Affinity DataIC50: 0.404nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716143(6-(((1S,2S,4S)-4-(2-chloro-5- (trifluoromethyl)phe...)
Affinity DataIC50: 0.409nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM715698(N-pyrimidin-4-yl-6-[rac- (1S,2S,4S)-2- (dimethylam...)
Affinity DataIC50: 0.427nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716126(5-fluoro-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2-(di...)
Affinity DataIC50: 0.427nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716150(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(4-fluoro-3- ...)
Affinity DataIC50: 0.473nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716160(2-methyl-6-(((1S,2S,4S)-2- morpholino-4-(3-(triflu...)
Affinity DataIC50: 0.527nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716132(5-chloro-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-4-(3-...)
Affinity DataIC50: 0.574nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716113(N-pyrimidin-4-yl-6-[[rac- (1S,2S,4S)-2-(dimethylam...)
Affinity DataIC50: 0.574nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716140(6-(((1S,2S,4S)-2-(cyclobutyl- (methyl)amino)-4-(3-...)
Affinity DataIC50: 0.597nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716122(N-pyrimidin-4-yl-6-[rac- (1S,2S,4S)-2-pyrrolidin-1...)
Affinity DataIC50: 0.602nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716144(6-(((1S,2S,4S)-4-(2,5-dichloro- phenyl)-2-(dimethy...)
Affinity DataIC50: 0.645nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716147(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(3-fluoro-5- ...)
Affinity DataIC50: 0.646nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716117(N-pyrimidin-4-yl-6-[rac- (1S,2S,4S)-4-[4-chloro-3-...)
Affinity DataIC50: 0.660nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716114(N-pyrimidin-4-yl-6-[rac- (1S,2S,4S)-2-pyrrolidin-1...)
Affinity DataIC50: 0.664nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716133(2-methyl-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2-(di...)
Affinity DataIC50: 0.664nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716148(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(2-fluoro-5- ...)
Affinity DataIC50: 0.687nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM715724(5-chloro-N-pyrimidin-4-yl-6- [[rac-(1S,2S,4S)-2- (...)
Affinity DataIC50: 0.765nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716128(2-methyl-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2-(di...)
Affinity DataIC50: 0.765nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716125(5-bromo-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2-(dim...)
Affinity DataIC50: 0.900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM715695(N-pyrimidin-4-yl-6-[rac- (1S,2S,4S)-2- (dimethylam...)
Affinity DataIC50: 0.900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716165(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(2-methyl-3- ...)
Affinity DataIC50: 0.909nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716151(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(2-fluoro-3- ...)
Affinity DataIC50: 0.917nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716162(6-(((1S,2S,4S)-4-(3-chloro- phenyl)-2-(dimethylami...)
Affinity DataIC50: 0.919nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716164(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(3-(2,2,2-tri...)
Affinity DataIC50: 0.942nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716158(6-(((1S,2S,4S)-2-(dimethyl- amino)-4-(3-(trifluoro...)
Affinity DataIC50: 0.989nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716168(6-(((1S,2S,4S)-2-(dimethy- lamino)-4-(3-((trifluor...)
Affinity DataIC50: 1.05nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716116(N-pyrimidin-4-yl-6-[[rac- (1S,2S,4S)-4-[4-chloro-3...)
Affinity DataIC50: 1.07nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716135(2-methyl-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2-pyr...)
Affinity DataIC50: 1.07nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716169(5-cyclopropyl-N-pyrimidin-4- yl-6-[rac-(1S,2S,4S)-...)
Affinity DataIC50: 1.16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716131(N-pyrimidin-4-yl-6-[rac- (1S,2S,4S)-2-(1-piperidyl...)
Affinity DataIC50: 1.16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716167(6-(((1S,2S,4S)-4-(5-chloro-6- (trifluoromethyl)pyr...)
Affinity DataIC50: 1.53nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716118(5-chloro-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2-(di...)
Affinity DataIC50: 1.55nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716152(6-(((1S,2S,4S)-2-(Diethy- lamino)-4-(3-(trifluoro-...)
Affinity DataIC50: 1.73nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716149(2-Chloro-6-(((1S,2S,4S)-2- (dimethylamino)-4-(2-fl...)
Affinity DataIC50: 1.81nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716157(6-(((1S,2S,4S)-4-(3-(difluoro- methoxy)phenyl)-2-(...)
Affinity DataIC50: 1.82nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716146(6-(((1S,2S,4S)-4-(3-(1,1- difluoroethyl)phenyl)-2-...)
Affinity DataIC50: 1.95nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM715721(5-chloro-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2- (d...)
Affinity DataIC50: 2.21nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716127(2-chloro-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2-(di...)
Affinity DataIC50: 2.21nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716121(N-pyrimidin-4-yl-6-[rac- (1S,2S,4S)-2-pyrrolidin-1...)
Affinity DataIC50: 2.79nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM716130(formic acid; N-pyrimidin-4-yl- 6-[rac-(1S,2S,4S)-2...)
Affinity DataIC50: 3.51nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM715733(5-cyano-N-pyrimidin-4-yl-6- [rac-(1S,2S,4S)-2- (di...)
Affinity DataIC50: 3.51nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
Go to US Patent

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