Compile Data Set for Download or QSAR
Report error Found 232 Enz. Inhib. hit(s) with all data for entry = 12535
LigandPNGBDBM709139(6-[5-({[3-(cyclobutylmeth-oxy)phenyl]methyl}carbam...)
Affinity DataIC50: 0.0400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709106(6-(5-{[(2-ethylphenyl)methyl]-carbamoyl}-6-methoxy...)
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709075(6-[6-methoxy-5-({[(1S,2R)-2-phenylcyclopropyl]meth...)
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709117(6-[6-methoxy-5-({[2-(propan-2-yloxy)phenyl]methyl}...)
Affinity DataIC50: 1.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709104(6-[6-methoxy-5-({[2-(propane-2-sulfonyl)phenyl]met...)
Affinity DataIC50: 1.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709161(6-[5-({[2-fluoro-5-(trifluoro-methoxy)phenyl]methy...)
Affinity DataIC50: 1.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709072(6-{6-methoxy-5-[(3-phenylbutyl)-carbamoyl]pyridin-...)
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709076(6-[6-methoxy-5-({[(1R,2S)-2-phenylcyclopropyl]meth...)
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709099(6-[6-methoxy-5-({[2-(2,2,2-trifluoroethoxy)phenyl]...)
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709103(6-(6-methoxy-5-{[(2-phenyl-oxan-3-yl)methyl]carbam...)
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709115(6-{5-[(2-{[(4-fluorophenyl)-methyl]carbamoyl}-2,2-...)
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709154(6-[5-({[5-fluoro-2-(propan-2-yloxy)phenyl]methyl}c...)
Affinity DataIC50: 1.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM707964(US12172975, Example 21-4)
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709181(6-[5-({[2-(cyclopentyloxy)-5-fluoro-phenyl]methyl}...)
Affinity DataIC50: 2.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM707954(6-(6-methoxy D3-5-((2-(trifluoromethoxy)benzyl D2)...)
Affinity DataIC50: 2.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709066(6-(5-{[(1R)-1-[2-fluoro-5-(tri-fluoromethyl)phenyl...)
Affinity DataIC50: 2.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709087(6-(5-{[3-(4-fluorophenoxy)-propyl]carbamoyl}-6-met...)
Affinity DataIC50: 2.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709151(6-[5-({[2-fluoro-6-(propan-2-yloxy)phenyl]methyl}-...)
Affinity DataIC50: 2.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709152(6-[5-({[2-(cyclopropylmeth-oxy)-3,5-difluorophenyl...)
Affinity DataIC50: 2.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709074(6-[5-({[4-fluoro-2-(oxan-4-yl-oxy)phenyl]methyl}ca...)
Affinity DataIC50: 2.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709110(6-[5-({[2-(cyclobutylmethoxy)-phenyl]methyl}carbam...)
Affinity DataIC50: 2.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709062(6-(5-{[(3S)-3-(4-chlorophenyl)-3-hydroxypropyl]car...)
Affinity DataIC50: 2.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709077(6-[6-methoxy-5-([2-(morpholin-4-yl)phenyl]methyl}c...)
Affinity DataIC50: 2.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709141(6-[5-({[3-(cyclobutylmethoxy)-pyridin-2-yl]methyl}...)
Affinity DataIC50: 2.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709102(6-[5-({[2-(difluoromethoxy)-phenyl]methyl}carbamoy...)
Affinity DataIC50: 2.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709116(6-[6-methoxy-5-({[3-(trifluoro-methoxy)phenyl]meth...)
Affinity DataIC50: 2.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709083(6-[6-methoxy-5-({[2-(2-meth-ylpropoxy)phenyl]methy...)
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709177(6-[6-methoxy-5-({[2-(trifluoro-methoxy)phenyl]{met...)
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709178(N-methyl-6-(6-methyl-5-{[(1S,3R)-3-phenylcyclopent...)
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709201(6-[6-methoxy-5-({[2-(trifluoro-methoxy)phenyl]meth...)
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709105(6-(5-{[(2,2-dimethylcyclo-hexyl)methyl]carbamoyl}-...)
Affinity DataIC50: 3.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709081(6-{5-[({2-[4-(hydroxymethyl)-piperidin-1-yl]phenyl...)
Affinity DataIC50: 3.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM707961(US12172975, Example 21-1)
Affinity DataIC50: 3.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM707948((S)-6-(5-((1-(2-fluoro-5-(trifluoromethoxy)phenyl)...)
Affinity DataIC50: 3.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709109(6-[5-({[2-(cyclopropylsulfam-oyl)phenyl]methyl}car...)
Affinity DataIC50: 3.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709180(N-methyl-6-[6-methyl-5-({1-[3-(tri-fluoromethoxy)p...)
Affinity DataIC50: 3.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709101(tert-butyl N-[(1R,2S)-2-[({2-methoxy-5-[3-(methylc...)
Affinity DataIC50: 3.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709111(6-(6-methoxy-5-{[3-(2,2,2-trifluoroethoxy)cyclohex...)
Affinity DataIC50: 3.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709239(6-(5-{[(1R)-1-[2-fluoro-5-(trifluoro-methyl)phenyl...)
Affinity DataIC50: 3.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM707944((R)-6-(5-((1-(2-fluoro-5-(trifluoromethyl)phenyl) ...)
Affinity DataIC50: 4.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709150(6-[5-({[3,5-difluoro-2-(propan-2-yloxy)phenyl]meth...)
Affinity DataIC50: 4.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709093(6-[6-methoxy-5-({[2-(propane-1-sulfonyl)phenyl]met...)
Affinity DataIC50: 4.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709125(6-[6-methoxy-5-({1-[3-(tri-fluoromethyl)phenyl]eth...)
Affinity DataIC50: 4.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709092(6-[6-methoxy-5-({[1-(phenoxy-methyl)cyclopropyl]me...)
Affinity DataIC50: 4.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709091(6-(6-methoxy-5-{[(1S,3R)-3-phenylcyclopentyl]carba...)
Affinity DataIC50: 4.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709097(tert-butyl-N-{2-[({2-methoxy-5-[3-(methylcarbamoyl...)
Affinity DataIC50: 4.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709136(6-[5-({[2-(cyclobutylmeth-oxy)pyridin-3-yl]methyl}...)
Affinity DataIC50: 4.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM707953(6-(6-methoxy d3-5-((1-(2-(trifluoromethoxy)phenyl)...)
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM709090(6-(5-{[(2-methanesulfonyl-phenyl)methyl]carbamoyl}...)
Ligand InfoPC cidPC sid
In DepthDetails

LigandPNGBDBM707967(4-fluoro-6-[6-methoxy-5-({1-[2-(trifluoromethoxy)p...)
Affinity DataIC50: 5.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

Displayed 1 to 50 (of 232 total ) | Next | Last >>
Jump to: