Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 11214
TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600774(US11633395, Example 18)
Affinity DataIC50: 6.90nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600771(US11633395, Example 15)
Affinity DataIC50: 7.80nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600769(US11633395, Example 13)
Affinity DataIC50: 7.90nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600770(US11633395, Example 14)
Affinity DataIC50: 9.10nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600758(US11633395, Example 2)
Affinity DataIC50: 11nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600763(US11633395, Example 7)
Affinity DataIC50: 11nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600772(US11633395, Example 16)
Affinity DataIC50: 13nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600775(US11633395, Example 19)
Affinity DataIC50: 16nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600768(US11633395, Example 12)
Affinity DataIC50: 16nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600773(US11633395, Example 17)
Affinity DataIC50: 17nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600761(US11633395, Example 5)
Affinity DataIC50: 18nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600757(US11633395, Example 1)
Affinity DataIC50: 18nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600764(US11633395, Example 8)
Affinity DataIC50: 19nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600759(US11633395, Example 3)
Affinity DataIC50: 23nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600762(US11633395, Example 6)
Affinity DataIC50: 26nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600760(US11633395, Example 4)
Affinity DataIC50: 33nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600765((7S)-5-[4-(difluoromethoxy)phenyl]-3-(imidazo[1,2-...)
Affinity DataIC50: 61nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600767(US11633395, Example 11)
Affinity DataIC50: 78nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
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TargetMetabotropic glutamate receptor 2(Human)
Sumitomo Pharma

US Patent
LigandPNGBDBM600766((7S)-5-[4-(trifluoromethyl)phenyl]-3-(2-aminoimida...)
Affinity DataIC50: 302nMAssay Description:Human mGlu2 receptor stable expressing cells were prepared and incubated. Luminescence signals by mGlu2 receptor stimulation were detected with FDSS7...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
Go to US Patent