Compile Data Set for Download or QSAR
Report error Found 211 Enz. Inhib. hit(s) with all data for entry = 11041
LigandPNGBDBM587697(5-(2-ethoxy-3-pyridyl)-N-ethyl-1-isopropyl- 3-meth...)
Affinity DataIC50: 5nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587713(2-(2-ethoxy-3-pyridyl)-8-methyl-6-[1- methylpropyl...)
Affinity DataIC50: 6nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587696(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N,3- dimethyl-p...)
Affinity DataIC50: 7nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587707((+-)-2-(2-ethoxy-3-pyridyl)-8-methyl-6-sec- butyl-...)
Affinity DataIC50: 9nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587698((+-)-5-[[[5-(2-ethoxy-3-pyridyl)-1-isopropyl- 3-me...)
Affinity DataIC50: 11nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587699(4-[[[5-(2-ethoxy-3-pyridyl)-1-isopropyl-3- methyl-...)
Affinity DataIC50: 12nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587700(5-(2-ethoxy-3-pyridyl)-1-isopropyl-3- methyl-pyraz...)
Affinity DataIC50: 13nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587694(5-(2-ethoxy-3-pyridyl)-1-isopropyl-3,6- dimethyl-p...)
Affinity DataIC50: 16nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587702(2-(2-ethoxy-3-pyridyl)-6-isopropyl-3,8- dimethyl-i...)
Affinity DataIC50: 17nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587695(1-isopropyl-3,6-dimethyl-5-(2-propoxy-3- pyridyl)p...)
Affinity DataIC50: 25nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587690(5-(2-ethoxy-3-pyridyl)-1-isopropyl-3- methyl-pyraz...)
Affinity DataIC50: 26nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587654(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N- [tetrahydrof...)
Affinity DataIC50: 32nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587714(2-(2-ethoxy-3-pyridyl)-8-methyl-6-[1- methylpropyl...)
Affinity DataIC50: 33nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587703(2-(2-ethoxy-3-pyridyl)-6-isopropyl-8- methyl-imida...)
Affinity DataIC50: 34nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587706(2-(2-ethoxy-3-pyridyl)-6-(1-ethylpropyl)-8- methyl...)
Affinity DataIC50: 36nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587653(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N- [tetrahydrof...)
Affinity DataIC50: 48nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587696(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N,3- dimethyl-p...)
Affinity DataIC50: 50nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587713(2-(2-ethoxy-3-pyridyl)-8-methyl-6-[1- methylpropyl...)
Affinity DataIC50: 51nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587690(5-(2-ethoxy-3-pyridyl)-1-isopropyl-3- methyl-pyraz...)
Affinity DataIC50: 52nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587699(4-[[[5-(2-ethoxy-3-pyridyl)-1-isopropyl-3- methyl-...)
Affinity DataIC50: 53nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587697(5-(2-ethoxy-3-pyridyl)-N-ethyl-1-isopropyl- 3-meth...)
Affinity DataIC50: 60nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587707((+-)-2-(2-ethoxy-3-pyridyl)-8-methyl-6-sec- butyl-...)
Affinity DataIC50: 61nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587700(5-(2-ethoxy-3-pyridyl)-1-isopropyl-3- methyl-pyraz...)
Affinity DataIC50: 62nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587698((+-)-5-[[[5-(2-ethoxy-3-pyridyl)-1-isopropyl- 3-me...)
Affinity DataIC50: 70nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587702(2-(2-ethoxy-3-pyridyl)-6-isopropyl-3,8- dimethyl-i...)
Affinity DataIC50: 74nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587713(2-(2-ethoxy-3-pyridyl)-8-methyl-6-[1- methylpropyl...)
Affinity DataIC50: 77nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587710(2-(2-ethoxy-3-pyridyl)-8-methyl-6-(oxetan- 3-yl)im...)
Affinity DataIC50: 78nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587594(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N- [trans-4-met...)
Affinity DataIC50: 82nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587583(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N- [[(2R)-tetra...)
Affinity DataIC50: 83nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587649(5-(2-ethoxy-3-pyridyl)-1-isopropyl-7- pyrrolidin-1...)
Affinity DataIC50: 83nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587692(1-isopropyl-5-(2-methoxy-3-pyridyl)-3,6- dimethyl-...)
Affinity DataIC50: 84nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587597(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N- methyl-pyraz...)
Affinity DataIC50: 85nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587651(5-(2-ethoxy-3-pyridyl)-1-ethyl-N- [tetrahydrofuran...)
Affinity DataIC50: 86nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587694(5-(2-ethoxy-3-pyridyl)-1-isopropyl-3,6- dimethyl-p...)
Affinity DataIC50: 86nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587699(4-[[[5-(2-ethoxy-3-pyridyl)-1-isopropyl-3- methyl-...)
Affinity DataIC50: 88nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587667(5-(2-tert-butoxy-3-pyridyl)-1-isopropyl-N- [(3R)-t...)
Affinity DataIC50: 91nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587569(5-(2-ethoxy-3-pyridyl)-1-(oxetan-3-yl)-7- pyrrolid...)
Affinity DataIC50: 95nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587703(2-(2-ethoxy-3-pyridyl)-6-isopropyl-8- methyl-imida...)
Affinity DataIC50: 96nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587701(5-(2-ethoxy-3-pyridyl)-1-isopropyl- pyrazolo[4,3-b...)
Affinity DataIC50: 99nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587702(2-(2-ethoxy-3-pyridyl)-6-isopropyl-3,8- dimethyl-i...)
Affinity DataIC50: 99nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587698((+-)-5-[[[5-(2-ethoxy-3-pyridyl)-1-isopropyl- 3-me...)
Affinity DataIC50: 106nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587596(5-(2-ethoxy-3-pyridyl)-N,1-diisopropyl- pyrazolo[4...)
Affinity DataIC50: 108nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587581(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N- [[(2S)-tetra...)
Affinity DataIC50: 111nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587696(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N,3- dimethyl-p...)
Affinity DataIC50: 111nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587707((+-)-2-(2-ethoxy-3-pyridyl)-8-methyl-6-sec- butyl-...)
Affinity DataIC50: 112nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587695(1-isopropyl-3,6-dimethyl-5-(2-propoxy-3- pyridyl)p...)
Affinity DataIC50: 118nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587704(6-cyclobutyl-2-(2-ethoxy-3-pyridyl)-8- methyl-imid...)
Affinity DataIC50: 121nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587691(1-isopropyl-3,6-dimethyl-5-phenyl- pyrazolo[4,3-b]...)
Affinity DataIC50: 122nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587660(1-isopropyl-5-(2-methoxy-3-pyridyl)-N- [(3R)-tetra...)
Affinity DataIC50: 124nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

LigandPNGBDBM587593(5-(2-ethoxy-3-pyridyl)-1-isopropyl-N- tetrahydropy...)
Affinity DataIC50: 126nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays were performed in 60 μL samples containing a fixed amount of the PDE1 enzyme...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent

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