Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 10934
TargetRho-associated protein kinase 2(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 8nMAssay Description:Table 2: ROCK-II(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-II(h) was in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 14nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 15nMAssay Description:Table 2: ROCK-II(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-II(h) was in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 15nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50156686(CHEMBL3794389 | US11485707, Example 23)
Affinity DataIC50: 17nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50156686(CHEMBL3794389 | US11485707, Example 23)
Affinity DataIC50: 17nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 18nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50156686(CHEMBL3794389 | US11485707, Example 23)
Affinity DataIC50: 18nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 18nMAssay Description:Table 2: ROCK-II(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-II(h) was in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 19nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 19nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 19nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 20nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50156686(CHEMBL3794389 | US11485707, Example 23)
Affinity DataIC50: 21nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50156686(CHEMBL3794389 | US11485707, Example 23)
Affinity DataIC50: 21nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 21nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 21nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 23nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 26nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 26nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50156686(CHEMBL3794389 | US11485707, Example 23)
Affinity DataIC50: 27nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 27nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 33nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50156686(CHEMBL3794389 | US11485707, Example 23)
Affinity DataIC50: 39nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 44nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Fochon Pharmaceuticals

US Patent
LigandPNGBDBM50546247(Netarsudil | AR-11324 FREE BASE | AR-13324 | US114...)
Affinity DataIC50: 64nMAssay Description:Table 2: ROCK-I(h) kinase assays were conducted using the KinaseProfiler service of Eurofins Pharma Discovery Services UK Limited. ROCK-I(h) was incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
Go to US Patent