Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 10825
TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571620(6-((5-(4-(1H-pyrazol-1- yl)phenyl)-1H-pyrazol-3- y...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571666(5-((5-(3-fluoro-4- hydroxyphenyl)-1H- pyrazol-3- y...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571674(6-((5-(4-(1H-imidazol-1- yl)phenyl)-1H-pyrazol-3- ...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571724(7-((5-(4-(1H-pyrazol-1- yl)phenyl)-1H-pyrazol-3- y...)
Affinity DataIC50: 7nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571722(4-(3-((1H-indazol-5- yl)amino)-1H-pyrazol-5- yl)ph...)
Affinity DataIC50: 29nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571723(4-(3-((1H-indazol-5- yl)amino)-1H-pyrazol-5- yl)-2...)
Affinity DataIC50: 45nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571721(N-(5-(4-(1H-pyrazol-1- yl)phenyl)-1H-pyrazol-3- yl...)
Affinity DataIC50: 55nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571612(6-((5-(4-hydroxyphenyl)- 1H-pyrazol-3-yl)amino)- 3...)
Affinity DataIC50: 62nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571553(N-(5-(4-methoxyphenyl)- 1H-pyrazol-3-yl)-1H- indaz...)
Affinity DataIC50: 94nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM571725(N-(5-(4-(1H-pyrazol-1- yl)phenyl)-1H-pyrazol-3- yl...)
Affinity DataIC50: 96nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11447469-20220920-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
Go to US Patent