Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 10791
TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569219(Step 1. 1-fluoro-N-methoxy-N-methylcyclobutane-1-c...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569210(US11427561, Compound 23)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569211(US11427561, Compound 24)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569212(US11427561, Compound 25)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569213(US11427561, Compound 26)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569214(US11427561, Compound 27)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569215(US11427561, Compound 28)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569216(US11427561, Compound 29)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569217(US11427561, Compound 30)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569218(Step 1. 1-fluoro-N-methoxy-N-methylcyclobutane-1-c...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569191(US11427561, Compound 2)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569220((R)-(6-(6-(6-(amino(3,3-difluorocyclobutyl)methyl)...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569221((S)-(6-(6-(6-(amino(3,3-difluorocyclobutyl)methyl)...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569222(US11427561, Compound 35a)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569200(US11427561, Compound 35b | (1R,3s)-3-((S)-amino(6-...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569224(US11427561, Compound 35c)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569225(US11427561, Compound 35d)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569226(US11427561, Compound 35i | US11427561, Compound 35...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569227(US11427561, Compound 35g)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569228(US11427561, Compound 35h)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569208(US11427561, Compound 21)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569190(US11427561, Compound 3 | (S)-(6-(6-(6-(amino(3-(hy...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569190(US11427561, Compound 3 | (S)-(6-(6-(6-(amino(3-(hy...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
Go to US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569193(US11427561, Compound 4)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569194((6-(6-(6-((R)-amino((cis-3-(tert-butyldimethylsily...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569195(trans-3-((S)-amino(6-(1-(6-(hydroxymethyl)pyridin-...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569196(trans-3-((R)-amino(6-(1-(6-(hydroxymethyl)pyridin-...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
Go to US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569197(US11427561, Compound 8)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569198(US11427561, Compound 9)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
Go to US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569199(US11427561, Compound 10)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569200(US11427561, Compound 35b | (1R,3s)-3-((S)-amino(6-...)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
Go to US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569201(US11427561, Compound 13)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
Go to US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569202(US11427561, Compound 14)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569203(US11427561, Compound 15)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
Go to US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569204(US11427561, Compound 16)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569205(US11427561, Compound 17)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569206(US11427561, Compound 19)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
Go to US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569207(US11427561, Compound 20)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
Go to US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569209(US11427561, Compound 22)
Affinity DataIC50: 100nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569229(US11427561, Compound 11)
Affinity DataIC50: 550nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569230(US11427561, Compound 18)
Affinity DataIC50: 550nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569231(US11427561, Compound 35e)
Affinity DataIC50: 550nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
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TargetInterleukin-1 receptor-associated kinase 4(Human)
Biogen Ma

US Patent
LigandPNGBDBM569226(US11427561, Compound 35i | US11427561, Compound 35...)
Affinity DataIC50: 550nMAssay Description:Biochemical Assay: The biochemical assay is in a AlphaScreen format. The kinase reaction is based on the IRAK-4 phosphorylation of a biotin labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
Go to US Patent