Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 10445
TargetCalpain-1 catalytic subunit(Human)
Landsteiner Genmed

US Patent
LigandPNGBDBM535882(US11242312, Example 3)
Affinity DataIC50: 0.00800nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2022
Entry Details
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TargetCalpain-1 catalytic subunit(Human)
Landsteiner Genmed

US Patent
LigandPNGBDBM535880(US11242312, Example 1)
Affinity DataIC50: 0.0300nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2022
Entry Details
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TargetCalpain-1 catalytic subunit(Human)
Landsteiner Genmed

US Patent
LigandPNGBDBM535881(US11242312, Example 2)
Affinity DataIC50: 2.20nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2022
Entry Details
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TargetCalpain-1 catalytic subunit(Human)
Landsteiner Genmed

US Patent
LigandPNGBDBM535883(US11242312, Example 4)
Affinity DataIC50: 7.10nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2022
Entry Details
Go to US Patent

TargetCalpain-1 catalytic subunit(Human)
Landsteiner Genmed

US Patent
LigandPNGBDBM535885(N-((S)-1-(((S)-4-(cyclopropylamino)-3,4-dioxo-1-ph...)
Affinity DataIC50: 110nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2022
Entry Details
Go to US Patent

TargetCalpain-1 catalytic subunit(Human)
Landsteiner Genmed

US Patent
LigandPNGBDBM535884(N-((S)-1-(((S)-4-(cyclopropylamino)-3,4-dioxo-1-ph...)
Affinity DataIC50: 255nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2022
Entry Details
Go to US Patent