Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 10330
TargetGlutaminase kidney isoform, mitochondrial(Human)
The Johns Hopkins University

US Patent
LigandPNGBDBM50178230(CHEMBL3814265 | US11191732, Example 5)
Affinity DataIC50: 80nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
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TargetGlutaminase kidney isoform, mitochondrial(Human)
The Johns Hopkins University

US Patent
LigandPNGBDBM528362(US11191732, Example 6)
Affinity DataIC50: 100nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
The Johns Hopkins University

US Patent
LigandPNGBDBM528363(US11191732, Example 7)
Affinity DataIC50: 100nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
The Johns Hopkins University

US Patent
LigandPNGBDBM50400072(CHEMBL2178396 | US11191732, Example 3)
Affinity DataIC50: 1.90E+3nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
The Johns Hopkins University

US Patent
LigandPNGBDBM108460(CHEMBL2178393 | US8604016, 17 | US9938267, Cmpd ID...)
Affinity DataIC50: 2.70E+3nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
The Johns Hopkins University

US Patent
LigandPNGBDBM50400050(CHEMBL2177757 | US8604016, 1 | US9938267, Cmpd ID ...)
Affinity DataIC50: 3.30E+3nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
The Johns Hopkins University

US Patent
LigandPNGBDBM50400050(CHEMBL2177757 | US8604016, 1 | US9938267, Cmpd ID ...)
Affinity DataIC50: 3.30E+3nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
The Johns Hopkins University

US Patent
LigandPNGBDBM50400063(CHEMBL2177744 | US11191732, Example 4)
Affinity DataIC50: 4.60E+3nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
The Johns Hopkins University

US Patent
LigandPNGBDBM50400049(CHEMBL2177758 | US11191732, Example 2)
Affinity DataIC50: 1.00E+5nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)