Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 9417
TargetAmine oxidase [copper-containing] 3(Human)
Eli Lilly

US Patent
LigandPNGBDBM385387((E)-3-Fluoro-2-[[2-(4-methoxy-1-piperidyl)pyrimidi...)
Affinity DataIC50: 12nMAssay Description:Amine oxidase activity of recombinant SSAO, MAOa, and MAOb isoforms are measured using the MAO-Glo assay kit from Promega (V1402). Test compounds (wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Eli Lilly

US Patent
LigandPNGBDBM385388((E)-3-Fluoro-2-[[2-[(3S)-3-methoxypyrrolidin-1-yl]...)
Affinity DataIC50: 32nMAssay Description:Amine oxidase activity of recombinant SSAO, MAOa, and MAOb isoforms are measured using the MAO-Glo assay kit from Promega (V1402). Test compounds (wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmine oxidase [copper-containing] 3(Human)
Eli Lilly

US Patent
LigandPNGBDBM385389((3 S)-1-[5-[(E)-2-(Aminomethyl)-3-fluoro-allyloxy]...)
Affinity DataIC50: 52nMAssay Description:Amine oxidase activity of recombinant SSAO, MAOa, and MAOb isoforms are measured using the MAO-Glo assay kit from Promega (V1402). Test compounds (wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent