Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 9052
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437710(US10597382, Example 1)
Affinity DataIC50: 5.5nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
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Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437726(US10597382, Example 6)
Affinity DataIC50: 5.5nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437770(US10597382, Example 13)
Affinity DataIC50: 5.5nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437775(US10597382, Example 14)
Affinity DataIC50: 5.5nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437711(US10597382, Example 2)
Affinity DataIC50: 55nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437720(US10597382, Example 4 | US10597382, Example 3)
Affinity DataIC50: 55nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437728(US10597382, Example 7)
Affinity DataIC50: 55nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437737(US10597382, Example 9)
Affinity DataIC50: 55nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437749(US10597382, Example 10)
Affinity DataIC50: 55nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437778(US10597382, Example 15)
Affinity DataIC50: 55nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437779(US10597382, Example 16)
Affinity DataIC50: 55nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437720(US10597382, Example 4 | US10597382, Example 3)
Affinity DataIC50: 550nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437729(US10597382, Example 8)
Affinity DataIC50: 550nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437756(US10597382, Example 11)
Affinity DataIC50: 550nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437759(US10597382, Example 12)
Affinity DataIC50: 550nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
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TargetMitogen-activated protein kinase kinase kinase 5(Human)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM437722(US10597382, Example 5)
Affinity DataIC50: 1.00E+3nMAssay Description:ASK1 kinase was from Thermofisher (Catalogue # PV4011), ATP was from Sigma (Catalogue # A7699), HTRF KinEASE Assay System was obtained from Cisbio (B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2020
Entry Details
Go to US Patent