Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 8913
Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM428840(US10544152, Cpd # 27)
Affinity DataEC50:  0.330nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM50076245(WAY-163909 | CHEMBL1628670 | US10544152, Cpd # 1)
Affinity DataEC50:  18.2nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM428842(US10544152, Cpd # 18 | US10544152, Cpd # 36)
Affinity DataEC50:  2.40nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM428843(US10544152, Cpd # 35)
Affinity DataEC50:  119nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM428844(US10544152, Cpd # 44)
Affinity DataEC50:  51.9nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM428845(US10544152, Cpd # 45)
Affinity DataEC50:  218nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM428846(US10544152, Cpd # 46)
Affinity DataEC50:  575nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM428842(US10544152, Cpd # 18 | US10544152, Cpd # 36)
Affinity DataEC50:  1.20nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM428848(US10544152, Cpd # 17)
Affinity DataEC50:  1.48E+3nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2C(Human)
University of Texas

US Patent
LigandPNGBDBM428849(US10544152, Cpd # 37)
Affinity DataEC50:  72.4nMAssay Description:Cell Lines and Cell Culture.The PathHunter U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
Go to US Patent