Compile Data Set for Download or QSAR
Report error Found 98 Enz. Inhib. hit(s) with all data for entry = 8883
LigandPNGBDBM426364(US10526325, Compound A40 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426340(US10526325, Compound A16)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
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LigandPNGBDBM426341(US10526325, Compound A17)
Affinity DataKd:  1.65E+3nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
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LigandPNGBDBM426342(US10526325, Compound A18 | US10829489, Compound A1...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426344(US10526325, Compound A20 | US10829489, Compound A2...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426346(US10526325, Compound A22 | US10829489, Compound A2...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426348(US10526325, Compound A24 | US10829489, Compound A2...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426352(US10526325, Compound A28 | US10829489, Compound A2...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426353(US10526325, Compound A29 | US10829489, Compound A2...)
Affinity DataKd:  1.65E+3nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426354(US10526325, Compound A30 | US10829489, Compound A3...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426356(US10526325, Compound A32 | US10829489, Compound A3...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426358(US10526325, Compound A34 | US10829489, Compound A3...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426361(US10526325, Compound A37 | US10829489, Compound A3...)
Affinity DataKd:  1.65E+3nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426362(US10526325, Compound A38 | US10829489, Compound A3...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426324(US10526325, Compound A1 | US10829489, Compound A1 ...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426366(US10526325, Compound A42 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426367(US10526325, Compound A43)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426368(US10526325, Compound A44 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426369(US10526325, Compound A45 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426370(US10526325, Compound A46 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426371(US10526325, Compound A47 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426372(US10526325, Compound A48 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426373(US10526325, Compound A49 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426374(US10526325, Compound A50 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
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Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426375(US10526325, Compound A51 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426376(US10526325, Compound A52 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426378(US10526325, Compound A54 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426381(US10526325, Compound A57 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426332(US10526325, Compound A9 | (2R)-1-[1-(4-chloropheny...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426331(US10526325, Compound A8 | US10829489, Compound A8 ...)
Affinity DataKd:  1.65E+3nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426330(US10526325, Compound A7 | US10829489, Compound A7 ...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426329(US10526325, Compound A6 | US10829489, Compound A6 ...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426328(US10526325, Compound A5 | US10829489, Compound A5 ...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426335(US10526325, Compound A12)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426334(US10526325, Compound A11 | US10829489, Compound A1...)
Affinity DataKd:  1.65E+3nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426327(US10526325, Compound A4 | US10829489, Compound A4 ...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426326(US10526325, Compound A3 | US10829489, Compound A3 ...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426337(US10526325, Compound A13)
Affinity DataKd:  1.65E+3nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426325(US10526325, Compound A2 | US10829489, Compound A2 ...)
Affinity DataKd:  1.65E+3nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426333(US10526325, Compound A10 | US10829489, Compound A1...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426338(US10526325, Compound A14 | US10829489, Compound A1...)
Affinity DataKd: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426356(US10526325, Compound A32 | US10829489, Compound A3...)
Affinity DataIC50: 300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426358(US10526325, Compound A34 | US10829489, Compound A3...)
Affinity DataIC50: 300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426333(US10526325, Compound A10 | US10829489, Compound A1...)
Affinity DataIC50: 300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426332(US10526325, Compound A9 | (2R)-1-[1-(4-chloropheny...)
Affinity DataIC50: 300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426362(US10526325, Compound A38 | US10829489, Compound A3...)
Affinity DataIC50: 300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426364(US10526325, Compound A40 | US10829489, Compound A4...)
Affinity DataIC50: 300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426330(US10526325, Compound A7 | US10829489, Compound A7 ...)
Affinity DataIC50: 300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426328(US10526325, Compound A5 | US10829489, Compound A5 ...)
Affinity DataIC50: 300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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LigandPNGBDBM426327(US10526325, Compound A4 | US10829489, Compound A4 ...)
Affinity DataIC50: 300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2020
Entry Details
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