Compile Data Set for Download or QSAR
Report error Found 120 Enz. Inhib. hit(s) with all data for entry = 8832
TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421947(US10494376, Example 55)
Affinity DataIC50: 16nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM422000(US10494376, Example 108)
Affinity DataIC50: 17nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421943(US10494376, Example 50)
Affinity DataIC50: 19nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421942(US10494376, Example 49)
Affinity DataIC50: 38nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421997(US10494376, Example 105)
Affinity DataIC50: 38nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421920(US10494376, Example 27)
Affinity DataIC50: 44nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421973(US10494376, Example 81)
Affinity DataIC50: 51nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421919(US10494376, Example 26)
Affinity DataIC50: 53nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421979(US10494376, Example 87)
Affinity DataIC50: 57nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421944(US10494376, Example 51)
Affinity DataIC50: 61nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421975(US10494376, Example 83)
Affinity DataIC50: 65nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421995(US10494376, Example 103)
Affinity DataIC50: 65nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421992(US10494376, Example 100)
Affinity DataIC50: 66nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421994(US10494376, Example 102)
Affinity DataIC50: 68nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421914(US10494376, Example 21)
Affinity DataIC50: 70nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM422011(US10494376, Example 124)
Affinity DataIC50: 70nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421954(US10494376, Example 62)
Affinity DataIC50: 102nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421953(US10494376, Example 61)
Affinity DataIC50: 104nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421993(US10494376, Example 101)
Affinity DataIC50: 104nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421930(US10494376, Example 37)
Affinity DataIC50: 105nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421974(US10494376, Example 82)
Affinity DataIC50: 106nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421962(US10494376, Example 70)
Affinity DataIC50: 121nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421983(US10494376, Example 91)
Affinity DataIC50: 123nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421976(US10494376, Example 84)
Affinity DataIC50: 124nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421991(US10494376, Example 99)
Affinity DataIC50: 127nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421923(US10494376, Example 30)
Affinity DataIC50: 139nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421996(US10494376, Example 104)
Affinity DataIC50: 147nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421929(US10494376, Example 36)
Affinity DataIC50: 148nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421928(US10494376, Example 35)
Affinity DataIC50: 152nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421972(US10494376, Example 80)
Affinity DataIC50: 161nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421971(US10494376, Example 79)
Affinity DataIC50: 168nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421921(US10494376, Example 28)
Affinity DataIC50: 180nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421980(US10494376, Example 88)
Affinity DataIC50: 187nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421941(US10494376, Example 48)
Affinity DataIC50: 192nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421981(US10494376, Example 89)
Affinity DataIC50: 203nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421924(US10494376, Example 31)
Affinity DataIC50: 204nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421935(US10494376, Example 42)
Affinity DataIC50: 212nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421998(US10494376, Example 106)
Affinity DataIC50: 212nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421939(US10494376, Example 46)
Affinity DataIC50: 230nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421990(US10494376, Example 98)
Affinity DataIC50: 230nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM422012(US10494376, Example 125)
Affinity DataIC50: 232nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421955(US10494376, Example 63)
Affinity DataIC50: 245nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421956(US10494376, Example 64)
Affinity DataIC50: 261nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421968(US10494376, Example 76)
Affinity DataIC50: 262nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421977(US10494376, Example 85)
Affinity DataIC50: 279nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421926(US10494376, Example 33)
Affinity DataIC50: 305nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421959(US10494376, Example 67)
Affinity DataIC50: 307nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421984(US10494376, Example 92)
Affinity DataIC50: 310nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421958(US10494376, Example 66)
Affinity DataIC50: 329nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM421966(US10494376, Example 74)
Affinity DataIC50: 338nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
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