Compile Data Set for Download or QSAR
Report error Found 215 Enz. Inhib. hit(s) with all data for entry = 8725
LigandPNGBDBM414902(US10435414, Compound 171 | (S)-2-((1-(2- aminobenz...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272899(BDBM414935 | US10065970, Compound 204 | (S)-2-((1-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272903((S)-2-((2-(2- aminobenzo[d]oxazol- 5-yl)-3,4-dihyd...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272865((S)-2-((1-(2- aminobenzo[d]thiazol- 6-yl)-8,9-dihy...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272936((S)-2-((1-(2-amino-4- fluorobenzo[d]oxazol- 5-yl)-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272937((S)-2-((1-(2-amino-4- fluorobenzo[d]thiazol- 6-yl)...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272938((S)-2-((1-(4-(1H- 1,2,4-triazol-3- yl)phenyl)-7,8,...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272939((S)-2-((1-(2- aminoquinoxalin-6- yl)-7,8,9,10- tet...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272941((S)-2-((1-(2- Aminobenzo[d]thiazol- 5-yl)-7,8,9,10...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272944((S)-2-((1-(2-amino-7- fluorobenzo[d]oxazol- 5-yl)-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272945((S)-1-(1-(2- aminobenzo[d]oxazol- 5-yl)-7,8,9,10- ...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272949((S)-2-((1-(2- aminobenzo[d]oxazol- 5-yl)-7,8,9,10-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272956((S)-2-((1-(2-amino-4,7- difluorobenzo[d]oxazol- 5-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272959((S)-2-((1-(2-amino-7- fluorobenzo[d]oxazol- 5-yl)-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272960((S)-2-((1-(2- aminothiazolo[5,4- b]pyridin-5-yl)- ...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272964((S)-2-((1-(3-fluoro-4- (1H-1,2,4-triazol-3- yl)phe...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272966((S)-2-((1-(2- aminobenzo[d]oxazol- 5-yl)-7,8,9,10-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272967((S)-2-((1-(2-amino-7- fluorobenzo[d]oxazol- 5-yl)-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272975((S)-2-((1-(2-amino-4- fluorobenzo[d]thiazol- 6-yl)...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272979((S)-2-((1-(2- aminobenzo[d]oxazol- 5-yl)-7,8,9,10-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272984((S)-2-((1-(2-amino-7- fluorobenzo[d]oxazol- 5-yl)-...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272989((2R,3S)-1-(1-(2- aminobenzo[d]oxazol- 5-yl)-7,8,9,...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272991((S)-2-((1-(5-(1H-1,2,4- triazol-5-yl)pyridin-2- yl...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM273000((S)-2-cyclopropyl-2- ((1-(3-fluoro-4-(1H- 1,2,4-tr...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM273002((S)-2-((1-(5-fluoro-6- (1H-1,2,4-triazol-5- yl)pyr...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM415047(US10435414, Example 315 | (S)-2-((1-(2- aminothiaz...)
Affinity DataKi: <0.0200nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272963((S)-2-((1-(4-(1H-1,2,4- triazol-3-yl)phenyl)- 7,8,...)
Affinity DataKi:  0.0210nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272988((S)-2-((1-(2-fluoro-4- (1H-1,2,4-triazol-5- yl)phe...)
Affinity DataKi:  0.0220nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM414979(US10435414, Example 247 | (S)-1-(1-(2- aminobenzo[...)
Affinity DataKi:  0.0240nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272987((S)-2-((1-(3- aminobenzo[e][1,2,4]tri- azin-7-yl)-...)
Affinity DataKi:  0.0240nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272889((S)-1-(1-(2- aminobenzo[d]oxazol- 5-yl)-3-fluoro-8...)
Affinity DataKi:  0.0260nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272976((S)-2-((1-(2- aminobenzo[d]thiazol- 6-yl)-7,8,9,10...)
Affinity DataKi:  0.0270nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272943((S)-2-((1-(2- aminobenzo[d]thiazol- 6-yl)-7,8,9,10...)
Affinity DataKi:  0.0300nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272965((S)-2-((1-(2-amino-4- fluorobenzo[d]oxazol- 5-yl)-...)
Affinity DataKi:  0.0300nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM415043(US10435414, Example 311 | (S)-2-(4-(1-(2- aminooxa...)
Affinity DataKi:  0.0310nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272800((S)-2-((1-(2- aminobenzo[d]oxazol- 5-yl)-8,9-dihyd...)
Affinity DataKi:  0.0320nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272940((R)-2-((1-(2- aminobenzo[d]oxazol- 5-yl)-7,8,9,10-...)
Affinity DataKi:  0.0320nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272934((S)-1-(1-(2- aminobenzo[d]thiazol- 6-yl)-7,8,9,10-...)
Affinity DataKi:  0.0350nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272996((S)-2-(4-(1-(2- aminooxazolo[4,5- b]pyridin-5-yl)-...)
Affinity DataKi:  0.0380nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM415044(US10435414, Example 312 | (R)-2-(4-(1-(2- aminooxa...)
Affinity DataKi:  0.0390nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM273003(US10065970, Example 309 | (2S,3S)-1-(1-(2- aminobe...)
Affinity DataKi:  0.0400nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272933((S)-2-(((R)-2-(2- aminobenzo[d]oxazol- 5-yl)-4-met...)
Affinity DataKi:  0.0450nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272995((2S,3R)-1-(1-(2- aminobenzo[d]thiazol- 6-yl)-7,8,9...)
Affinity DataKi:  0.0450nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272968((S)-2-((1-(2-amino-4- fluorobenzo[d]thiazol- 6-yl)...)
Affinity DataKi:  0.0490nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272990((S)-2-((1-(2,5-difluoro- 4-(1H-1,2,4-triazol-5- yl...)
Affinity DataKi:  0.0530nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272882((S)-2-((1-(2- aminoquinoxalin-6- yl)-8,9-dihydro-7...)
Affinity DataKi:  0.0560nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272994((R)-2-(4-(1-(2- aminothiazolo[5,4- b]pyridin-5-yl)...)
Affinity DataKi:  0.0610nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272980((S)-2-((1-(2-amino-7- fluorobenzo[d]thiazol- 5-yl)...)
Affinity DataKi:  0.0620nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272993((S)-2-(4-(1-(2- aminothiazolo[5,4- b]pyridin-5-yl)...)
Affinity DataKi:  0.0700nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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LigandPNGBDBM272799((S)-1-(1-(2- aminobenzo[d]oxazol- 5-yl)-8,9-dihydr...)
Affinity DataKi:  0.0710nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
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