Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 8666
TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)
Affinity DataIC50: 2.80nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)
Affinity DataIC50: 3.30nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412135(US10392402, Compound ID 52 | US10807966, Compound ...)
Affinity DataIC50: 8.70nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412127(US10392402, Compound ID 5 | US10807966, Compound 2...)
Affinity DataIC50: 16.1nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412132(US10392402, Compound ID 40 | US10807966, Compound ...)
Affinity DataIC50: 17.4nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412130(US10392402, Compound ID 11 | US10807966, Compound ...)
Affinity DataIC50: 22.1nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412128(US10392402, Compound ID 7 | US10807966, Compound 7)
Affinity DataIC50: 22.9nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412131(US10392402, Compound ID 25)
Affinity DataIC50: 28.7nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412135(US10392402, Compound ID 52 | US10807966, Compound ...)
Affinity DataIC50: 34nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412129(US10392402, Compound ID 9 | US10807966, Compound 9)
Affinity DataIC50: 39.1nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412130(US10392402, Compound ID 11 | US10807966, Compound ...)
Affinity DataIC50: 63.6nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412132(US10392402, Compound ID 40 | US10807966, Compound ...)
Affinity DataIC50: 65.1nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412127(US10392402, Compound ID 5 | US10807966, Compound 2...)
Affinity DataIC50: 73nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412126(US10392402, Compound ID 1)
Affinity DataIC50: 98nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412128(US10392402, Compound ID 7 | US10807966, Compound 7)
Affinity DataIC50: 102nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412131(US10392402, Compound ID 25)
Affinity DataIC50: 130nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412126(US10392402, Compound ID 1)
Affinity DataIC50: 207nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412129(US10392402, Compound ID 9 | US10807966, Compound 9)
Affinity DataIC50: 237nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412134(US10392402, Compound ID 50)
Affinity DataIC50: 239nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412134(US10392402, Compound ID 50)
Affinity DataIC50: 1.01E+3nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412133(US10392402, Compound ID 48)
Affinity DataIC50: 1.87E+3nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412133(US10392402, Compound ID 48)
Affinity DataIC50: 6.40E+3nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/20/2020
Entry Details
Go to US Patent