Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 1378
LigandPNGBDBM318958(US10173995, Compound 2 | N-(5-(2,6-dimorpholinopyr...)
Affinity DataIC50: 0.400nMAssay Description:An in vitro assay which determines the ability of a test compound to inhibit PI3K alpha activity: PI3 alpha (PIK3CA) kinase-tagged T7 phage strains w...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM319549(US10173995, Compound 9)
Affinity DataIC50: 0.840nMAssay Description:An in vitro assay which determines the ability of a test compound to inhibit PI3K alpha activity: PI3 alpha (PIK3CA) kinase-tagged T7 phage strains w...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM318959(US10173995, Compound 4 | 5-(2,6-dimorpholinopyrimi...)
Affinity DataIC50: 1.90nMAssay Description:An in vitro assay which determines the ability of a test compound to inhibit PI3K alpha activity: PI3 alpha (PIK3CA) kinase-tagged T7 phage strains w...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM318960(US10173995, Compound 5 | 5-(2,6-dimorpholinopyrimi...)
Affinity DataIC50: 10nMAssay Description:An in vitro assay which determines the ability of a test compound to inhibit PI3K alpha activity: PI3 alpha (PIK3CA) kinase-tagged T7 phage strains w...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM318958(US10173995, Compound 2 | N-(5-(2,6-dimorpholinopyr...)
Affinity DataIC50: 32nMAssay Description:An in vitro assay which determines the ability of a test compound to inhibit PI3K alpha activity: PI3 delta (PIK3CD) kinase-tagged T7 phage strains w...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM319548(US10173995, Compound 6)
Affinity DataIC50: 60nMAssay Description:An in vitro assay which determines the ability of a test compound to inhibit PI3K alpha activity: PI3 alpha (PIK3CA) kinase-tagged T7 phage strains w...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50380363(CHEMBL2017974 | US10173995, Compound 1)
Affinity DataIC50: 310nMAssay Description:An in vitro assay which determines the ability of a test compound to inhibit PI3K alpha activity: PI3 delta (PIK3CD) kinase-tagged T7 phage strains w...More data for this Ligand-Target Pair
In DepthDetails
US Patent