Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 764
TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77055(US9694018, 8 | US10093697, 8. | US10487111, Exampl...)
Affinity DataIC50: 0.110nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77086(US9694018, 13 | US10093697, 13. | US10487111, Exam...)
Affinity DataIC50: 0.130nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77080(US9694018, 11 | US10093697, 11.)
Affinity DataIC50: 0.150nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77040(US9694018, 5 | US10093697, 5. | US10487111, Exampl...)
Affinity DataIC50: 0.160nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77029(US9694018, 3 | US10093697, 3. | US10487111, Exampl...)
Affinity DataIC50: 0.180nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77074(US9694018, 10 | US10093697, 10. | US10487111, Exam...)
Affinity DataIC50: 0.200nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77083(US9694018, 12 | US10093697, 12. | US10487111, Exam...)
Affinity DataIC50: 0.300nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77033(US9694018, 4 | US10093697, 4. | US10487111, Exampl...)
Affinity DataIC50: 0.350nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77051(US9694018, 7 | US10093697, 7. | US10487111, Exampl...)
Affinity DataIC50: 0.360nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
Go to US Patent

TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77074(US9694018, 10 | US10093697, 10. | US10487111, Exam...)
Affinity DataIC50: 0.390nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM76994(US9694018, 1 | US10093697, 1. | US10487111, Exampl...)
Affinity DataIC50: 0.450nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
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TargetIleal sodium/bile acid cotransporter(Human)
TBA

US Patent
LigandPNGBDBM77088(US9694018, 14 | US10093697, 14. | US10487111, Exam...)
Affinity DataIC50: 1.20nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2019
Entry Details
Go to US Patent