Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 3458
TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234465(US9353084, 18 | US10004738, 18)
Affinity DataKi:  4.30nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234464(US9353084, 17 | US10004738, 48)
Affinity DataKi:  11nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234451(US9353084, 4 | US10004738, 4)
Affinity DataKi:  11nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234450(US9353084, 3 | US10004738, 3)
Affinity DataKi:  12nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234464(US9353084, 17 | US10004738, 48)
Affinity DataKi:  14nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234492(US9353084, 46 | US10004738, 46)
Affinity DataKi:  14nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234491(US9353084, 45 | US10004738, 45)
Affinity DataKi:  14nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234452(US9353084, 5 | US10004738, 5)
Affinity DataKi:  18nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234453(US9353084, 6 | US10004738, 6)
Affinity DataKi:  19nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234460(US9353084, 13 | US10004738, 13)
Affinity DataKi:  28nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234459(US9353084, 12 | US10004738, 12)
Affinity DataKi:  29nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234466(US9353084, 19 | US10004738, 19)
Affinity DataKi:  32nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234454(US9353084, 7 | US10004738, 7)
Affinity DataKi:  33nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234461(US9353084, 14 | US10004738, 14)
Affinity DataKi:  37nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234457(US9353084, 10 | US10004738, 10)
Affinity DataKi:  44nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234462(US9353084, 15 | US10004738, 15)
Affinity DataKi:  46nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234479(US9353084, 32 | US10004738, 32)
Affinity DataKi:  51nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234463(US9353084, 16 | US10004738, 16)
Affinity DataKi:  58nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234468(US9353084, 21 | US10004738, 21)
Affinity DataKi:  58nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234494(US9353084, 49 | US10004738, 49)
Affinity DataKi:  60nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234480(US9353084, 33 | US10004738, 33)
Affinity DataKi:  62nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234458(US9353084, 11 | US10004738, 11)
Affinity DataKi:  63nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234493(US9353084, 47 | US10004738, 47)
Affinity DataKi:  65nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234455(US9353084, 8 | US10004738, 8)
Affinity DataKi:  66nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234470(US9353084, 23 | US10004738, 23)
Affinity DataKi:  71nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234448(US9353084, 1 | US10004738, 1)
Affinity DataKi:  83nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM401022(US10004738, 43 | N-(3-((2R,5R)-6-amino-3,3,5-trifl...)
Affinity DataKi:  91nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234476(US9353084, 29 | US10004738, 29)
Affinity DataKi:  92nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234478(US9353084, 31 | US10004738, 31)
Affinity DataKi:  92nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234456(US9353084, 9 | US10004738, 9)
Affinity DataKi:  100nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234469(US9353084, 22 | US10004738, 22)
Affinity DataKi:  110nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234472(US9353084, 25 | US10004738, 25)
Affinity DataKi:  130nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234473(US9353084, 26 | US10004738, 26)
Affinity DataKi:  130nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234474(US9353084, 27 | US10004738, 27)
Affinity DataKi:  140nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234475(US9353084, 28 | US10004738, 28)
Affinity DataKi:  170nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234481(US9353084, 34 | US10004738, 34)
Affinity DataKi:  210nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234449(US9353084, 2 | US10004738, 2)
Affinity DataKi:  210nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234477(US9353084, 30 | US10004738, 30)
Affinity DataKi:  260nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234483(US9353084, 36 | US10004738, 36)
Affinity DataKi:  390nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234484(US9353084, 37 | US10004738, 37)
Affinity DataKi:  420nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234471(US9353084, 24 | US10004738, 24)
Affinity DataKi:  420nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234488(US9353084, 41 | US10004738, 41)
Affinity DataKi:  520nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234482(US9353084, 35 | US10004738, 35)
Affinity DataKi:  680nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234490(US9353084, 44 | US10004738, 44)
Affinity DataKi:  740nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234485(US9353084, 38 | US10004738, 38)
Affinity DataKi:  1.00E+3nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234489(US9353084, 42 | US10004738, 42)
Affinity DataKi:  1.50E+3nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234467(US9353084, 20 | US10004738, 20)
Affinity DataKi:  1.60E+3nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234486(US9353084, 39 | US10004738, 39)
Affinity DataKi:  4.80E+3nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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TargetBeta-secretase 1(Human)
H. Lundbeck

US Patent
LigandPNGBDBM234487(US9353084, 40 | US10004738, 40)
Affinity DataKi:  8.20E+3nMAssay Description:The binding assay was performed as SPA-based assay using a biotinylated form of human BACE1 recombinantly expressed and subsequently purified from Fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
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