Compile Data Set for Download or QSAR
Report error Found 111 Enz. Inhib. hit(s) with all data for entry = 50008381
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072840(N-[1-(4-Diaminomethyl-benzyl)-2-oxo-2-piperidin-1-...)
Affinity DataKi:  6nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060033(3-[3-(4-Methyl-piperidin-1-yl)-2-(naphthalene-2-su...)
Affinity DataKi:  6.20nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072851(1-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  8.40nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072843(2,7-Bis-(4-diaminomethyl-benzylidene)-cycloheptano...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against bovine coagulation factor X expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072846(3-[3-(4-Methyl-piperidin-1-yl)-2-(naphthalene-1-su...)
Affinity DataKi:  16nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072854(1-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  17nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072856(3-[3-(4-Methyl-piperidin-1-yl)-3-oxo-2-(toluene-4-...)
Affinity DataKi:  26nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072847(3-[2-(9,10-Dioxo-9,10-dihydro-anthracene-2-sulfony...)
Affinity DataKi:  26nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060047(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-(4-phen...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTissue-type plasminogen activator(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072843(2,7-Bis-(4-diaminomethyl-benzylidene)-cycloheptano...)
Affinity DataKi:  35nMAssay Description:Inhibitory activity against human tissue-type plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072854(1-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  36nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072853(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  37nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072859(3-[3-(4-Methyl-piperidin-1-yl)-3-oxo-2-(2,4,6-trim...)
Affinity DataKi:  59nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060049(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-piperid...)
Affinity DataKi:  65nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072847(3-[2-(9,10-Dioxo-9,10-dihydro-anthracene-2-sulfony...)
Affinity DataKi:  74nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072857(3-[3-(4-Methyl-piperidin-1-yl)-3-oxo-2-(2,4,6-trii...)
Affinity DataKi:  75nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072843(2,7-Bis-(4-diaminomethyl-benzylidene)-cycloheptano...)
Affinity DataKi:  90nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072858(3-[3-(3-Methyl-piperidin-1-yl)-2-(naphthalene-2-su...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060033(3-[3-(4-Methyl-piperidin-1-yl)-2-(naphthalene-2-su...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072850(1-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072852(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  200nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060043(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-piperaz...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072851(1-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072841(3-(3-Diaminomethyl-phenyl)-2-[2-(naphthalene-2-sul...)
Affinity DataKi:  240nMAssay Description:Inhibitory activity against bovine coagulation factor X expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072843(2,7-Bis-(4-diaminomethyl-benzylidene)-cycloheptano...)
Affinity DataKi:  320nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060049(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-piperid...)
Affinity DataKi:  330nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072842(N-[1-(3-Diaminomethyl-benzyl)-2-oxo-2-piperidin-1-...)
Affinity DataKi:  340nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072850(1-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  390nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072853(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  410nMAssay Description:Inhibitory activity against human urokinase plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072855(1-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  460nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072853(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  490nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060043(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-piperaz...)
Affinity DataKi:  500nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060047(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-(4-phen...)
Affinity DataKi:  520nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072856(3-[3-(4-Methyl-piperidin-1-yl)-3-oxo-2-(toluene-4-...)
Affinity DataKi:  520nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072858(3-[3-(3-Methyl-piperidin-1-yl)-2-(naphthalene-2-su...)
Affinity DataKi:  530nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTissue-type plasminogen activator(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072853(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  570nMAssay Description:Inhibitory activity against human tissue-type plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072846(3-[3-(4-Methyl-piperidin-1-yl)-2-(naphthalene-1-su...)
Affinity DataKi:  630nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072840(N-[1-(4-Diaminomethyl-benzyl)-2-oxo-2-piperidin-1-...)
Affinity DataKi:  690nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072857(3-[3-(4-Methyl-piperidin-1-yl)-3-oxo-2-(2,4,6-trii...)
Affinity DataKi:  690nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072845(3-(3-Diaminomethyl-phenyl)-2-[2-(toluene-4-sulfony...)
Affinity DataKi:  840nMAssay Description:Inhibitory activity against bovine coagulation factor X expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTissue-type plasminogen activator(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072852(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  950nMAssay Description:Inhibitory activity against human tissue-type plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTissue-type plasminogen activator(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072855(1-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  980nMAssay Description:Inhibitory activity against human tissue-type plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072852(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072844([1-(3-Carbamimidoyl-benzyl)-2-(4-methyl-piperidin-...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072841(3-(3-Diaminomethyl-phenyl)-2-[2-(naphthalene-2-sul...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072842(N-[1-(3-Diaminomethyl-benzyl)-2-oxo-2-piperidin-1-...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072852(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibitory activity against human urokinase plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072855(1-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibitory activity against human urokinase plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072853(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibitory activity against bovine coagulation factor X expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072855(1-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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