Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50008069
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070439(2-{(S)-2-[(S)-2-(3,3-Dimethyl-butyrylamino)-3,3-di...)
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutrophil elastase(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070444((3R,4S)-3-Methyl-2-oxo-4-(pyridin-2-ylmethylsulfan...)
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against human leukocyte elastase protease(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070446(((S)-2,2-Dimethyl-1-{(S)-3-methyl-1-[4-oxo-1-((S)-...)
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070440({(S)-1-[(S)-1-(1-Benzylcarbamoyl-4-oxo-azetidin-2-...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070444((3R,4S)-3-Methyl-2-oxo-4-(pyridin-2-ylmethylsulfan...)
Affinity DataIC50: 730nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070440({(S)-1-[(S)-1-(1-Benzylcarbamoyl-4-oxo-azetidin-2-...)
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070438(2-Oxo-4-(2-oxo-2-phenyl-ethylsulfanyl)-azetidine-1...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070435(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070442({(S)-1-[(S)-1-(1-Benzylcarbamoyl-4-oxo-azetidin-2-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070443(((S)-2,2-Dimethyl-1-{(S)-3-methyl-1-[4-oxo-1-((R)-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070444((3R,4S)-3-Methyl-2-oxo-4-(pyridin-2-ylmethylsulfan...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50065878(2-Oxo-4-phenylsulfanyl-azetidine-1-carboxylic acid...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070441(2-Oxo-4-(pyridin-3-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070447(2-Oxo-4-(pyridin-4-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070448(2-Benzylsulfanyl-4-oxo-azetidine-1-carboxylic acid...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070445(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070449(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50065878(2-Oxo-4-phenylsulfanyl-azetidine-1-carboxylic acid...)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070436(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCapsid scaffolding protein(HHV-5)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070437(2-Oxo-4-phenethylsulfanyl-azetidine-1-carboxylic a...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibitory activity against human cytomegalovirus (HCMV) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070442({(S)-1-[(S)-1-(1-Benzylcarbamoyl-4-oxo-azetidin-2-...)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070447(2-Oxo-4-(pyridin-4-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070435(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070436(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070441(2-Oxo-4-(pyridin-3-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070449(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070434({4-[4-Oxo-1-((R)-1-phenyl-ethylcarbamoyl)-azetidin...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50065878(2-Oxo-4-phenylsulfanyl-azetidine-1-carboxylic acid...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070449(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070448(2-Benzylsulfanyl-4-oxo-azetidine-1-carboxylic acid...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070436(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070443(((S)-2,2-Dimethyl-1-{(S)-3-methyl-1-[4-oxo-1-((R)-...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070442({(S)-1-[(S)-1-(1-Benzylcarbamoyl-4-oxo-azetidin-2-...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutrophil elastase(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070445(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against human leukocyte elastase protease(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070447(2-Oxo-4-(pyridin-4-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070439(2-{(S)-2-[(S)-2-(3,3-Dimethyl-butyrylamino)-3,3-di...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070443(((S)-2,2-Dimethyl-1-{(S)-3-methyl-1-[4-oxo-1-((R)-...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutrophil elastase(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070434({4-[4-Oxo-1-((R)-1-phenyl-ethylcarbamoyl)-azetidin...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against human leukocyte elastase protease(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070445(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase(PPE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070446(((S)-2,2-Dimethyl-1-{(S)-3-methyl-1-[4-oxo-1-((S)-...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutrophil elastase(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070438(2-Oxo-4-(2-oxo-2-phenyl-ethylsulfanyl)-azetidine-1...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against human leukocyte elastase protease(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070449(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutrophil elastase(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070442({(S)-1-[(S)-1-(1-Benzylcarbamoyl-4-oxo-azetidin-2-...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against human leukocyte elastase protease(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutrophil elastase(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070449(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against human leukocyte elastase protease(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutrophil elastase(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070436(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against human leukocyte elastase protease(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutrophil elastase(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070435(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against human leukocyte elastase protease(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070434({4-[4-Oxo-1-((R)-1-phenyl-ethylcarbamoyl)-azetidin...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070446(((S)-2,2-Dimethyl-1-{(S)-3-methyl-1-[4-oxo-1-((S)-...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChymotrypsinogen B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070435(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50070437(2-Oxo-4-phenethylsulfanyl-azetidine-1-carboxylic a...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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