Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50008053
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070340(Thiophene-2-sulfonic acid [2-(3-{[((E)-6,6-dimethy...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070340(Thiophene-2-sulfonic acid [2-(3-{[((E)-6,6-dimethy...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of cholesterol biosynthesis in human HepG2 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070340(Thiophene-2-sulfonic acid [2-(3-{[((E)-6,6-dimethy...)
Affinity DataIC50: 80nMAssay Description:In vitro inhibition of dog liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070344(Thiophene-2-sulfonic acid [2-(3-{[((E)-6,6-dimethy...)
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070337([3,3']Bithiophenyl-5-sulfonic acid [2-(3-{[((E)-6,...)
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070341(Pyridine-3-sulfonic acid [2-(3-{[((E)-6,6-dimethyl...)
Affinity DataIC50: 150nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070343(Thiazole-2-sulfonic acid [2-(3-{[((E)-6,6-dimethyl...)
Affinity DataIC50: 170nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070345(Thiophene-2-sulfonic acid [2-(3-{[((E)-6,6-dimethy...)
Affinity DataIC50: 170nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070331(4-Cyano-N-[2-(3-{[((E)-6,6-dimethyl-hept-2-en-4-yn...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070350(N-[2-(3-{[((E)-6,6-Dimethyl-hept-2-en-4-ynyl)-ethy...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070346([2,3']Bithiophenyl-5-sulfonic acid [2-(3-{[((E)-6,...)
Affinity DataIC50: 210nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070342(Thiophene-2-sulfonic acid cyclopropyl-[2-(3-{[((E)...)
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070349(Thiophene-3-sulfonic acid [2-(3-{[((E)-6,6-dimethy...)
Affinity DataIC50: 250nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070333(N-[2-(3-{[((E)-6,6-Dimethyl-hept-2-en-4-ynyl)-ethy...)
Affinity DataIC50: 255nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070348(((E)-6,6-Dimethyl-hept-2-en-4-ynyl)-ethyl-{3-[3-(t...)
Affinity DataIC50: 290nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070339(4-Bromo-thiophene-2-sulfonic acid [2-(3-{[((E)-6,6...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070347(4-Bromo-N-[2-(3-{[((E)-6,6-dimethyl-hept-2-en-4-yn...)
Affinity DataIC50: 330nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070338(5-Bromo-thiophene-2-sulfonic acid [2-(3-{[((E)-6,6...)
Affinity DataIC50: 390nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070335(Thiophene-2-sulfonic acid [2-(3-{[((E)-6,6-dimethy...)
Affinity DataIC50: 450nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070334(Benzo[b]thiophene-2-sulfonic acid [2-(3-{[((E)-6,6...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070340(Thiophene-2-sulfonic acid [2-(3-{[((E)-6,6-dimethy...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibition of rat liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070336(Thiophene-2-sulfonic acid [3-(3-{[((E)-6,6-dimethy...)
Affinity DataIC50: 6.40E+3nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSqualene monooxygenase(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50070332([2,2']Bithiophenyl-5-sulfonic acid [2-(3-{[((E)-6,...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of pig liver squalene epoxidase in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed